Compile Data Set for Download or QSAR
maximum 50k data
Found 15 Enz. Inhib. hit(s) with all data for entry = 5723
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

LigandPNGBDBM92873(4-Aminoquinazoline derivative, 6h)
Affinity DataIC50:  62nMAssay Description:The kinase assay of Aurora A and B was measured using HTRF-kinEASE-STK discovery kit purchased from Cisbio.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

LigandPNGBDBM92870(4-Aminoquinazoline derivative, 6d)
Affinity DataIC50:  77nMAssay Description:The kinase assay of Aurora A and B was measured using HTRF-kinEASE-STK discovery kit purchased from Cisbio.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

LigandPNGBDBM92869(4-Aminoquinazoline derivative, 6c)
Affinity DataIC50:  98nMAssay Description:The kinase assay of Aurora A and B was measured using HTRF-kinEASE-STK discovery kit purchased from Cisbio.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

LigandPNGBDBM92871(4-Aminoquinazoline derivative, 6f)
Affinity DataIC50:  111nMAssay Description:The kinase assay of Aurora A and B was measured using HTRF-kinEASE-STK discovery kit purchased from Cisbio.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Southeast University

LigandPNGBDBM92871(4-Aminoquinazoline derivative, 6f)
Affinity DataIC50:  136nMAssay Description:The kinase assay of Aurora A and B was measured using HTRF-kinEASE-STK discovery kit purchased from Cisbio.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Southeast University

LigandPNGBDBM92870(4-Aminoquinazoline derivative, 6d)
Affinity DataIC50:  145nMAssay Description:The kinase assay of Aurora A and B was measured using HTRF-kinEASE-STK discovery kit purchased from Cisbio.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Southeast University

LigandPNGBDBM92873(4-Aminoquinazoline derivative, 6h)
Affinity DataIC50:  146nMAssay Description:The kinase assay of Aurora A and B was measured using HTRF-kinEASE-STK discovery kit purchased from Cisbio.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

LigandPNGBDBM92867(4-Aminoquinazoline derivative, 6a)
Affinity DataIC50:  179nMAssay Description:The kinase assay of Aurora A and B was measured using HTRF-kinEASE-STK discovery kit purchased from Cisbio.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Southeast University

LigandPNGBDBM92867(4-Aminoquinazoline derivative, 6a)
Affinity DataIC50:  191nMAssay Description:The kinase assay of Aurora A and B was measured using HTRF-kinEASE-STK discovery kit purchased from Cisbio.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Southeast University

LigandPNGBDBM92869(4-Aminoquinazoline derivative, 6c)
Affinity DataIC50:  202nMAssay Description:The kinase assay of Aurora A and B was measured using HTRF-kinEASE-STK discovery kit purchased from Cisbio.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

LigandPNGBDBM92868(4-Aminoquinazoline derivative, 6b)
Affinity DataIC50:  323nMAssay Description:The kinase assay of Aurora A and B was measured using HTRF-kinEASE-STK discovery kit purchased from Cisbio.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Southeast University

LigandPNGBDBM92868(4-Aminoquinazoline derivative, 6b)
Affinity DataIC50:  489nMAssay Description:The kinase assay of Aurora A and B was measured using HTRF-kinEASE-STK discovery kit purchased from Cisbio.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

LigandPNGBDBM92874(4-Aminoquinazoline derivative, 6i)
Affinity DataIC50:  788nMAssay Description:The kinase assay of Aurora A and B was measured using HTRF-kinEASE-STK discovery kit purchased from Cisbio.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

LigandPNGBDBM92872(4-Aminoquinazoline derivative, 6g)
Affinity DataIC50:  822nMAssay Description:The kinase assay of Aurora A and B was measured using HTRF-kinEASE-STK discovery kit purchased from Cisbio.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Southeast University

LigandPNGBDBM92874(4-Aminoquinazoline derivative, 6i)
Affinity DataIC50:  893nMAssay Description:The kinase assay of Aurora A and B was measured using HTRF-kinEASE-STK discovery kit purchased from Cisbio.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed