Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50042566
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50396238(CHEMBL2172212 | US9402842, 62)
Affinity DataEC50:  4.40E+3nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427892(CHEMBL2322286)
Affinity DataEC50:  1.84E+4nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50425045(CHEMBL2312896 | CHEMBL2322964 | US9402842, 43)
Affinity DataEC50:  8.40E+3nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50388545(CHEMBL1181674 | CHEMBL188130)
Affinity DataEC50:  1.59E+4nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50388546(CHEMBL213072 | CHEMBL333363)
Affinity DataEC50:  8.66E+3nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50388547(CHEMBL1181663 | CHEMBL187863)
Affinity DataEC50:  1.13E+4nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50388548(CHEMBL1182248 | CHEMBL225093)
Affinity DataEC50:  1.22E+4nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50388549(CHEMBL1185123 | CHEMBL390611)
Affinity DataEC50:  1.64E+4nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427893(CHEMBL2322288)
Affinity DataEC50:  1.07E+4nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427894(CHEMBL425544)
Affinity DataEC50:  9.60E+3nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427895(CHEMBL2322955)
Affinity DataEC50:  9.22E+3nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427896(CHEMBL2326683)
Affinity DataEC50:  7.00E+3nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50396236(CHEMBL2172210)
Affinity DataEC50:  1.52E+4nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50425054(CHEMBL2312904)
Affinity DataEC50: >2.07E+4nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50396234(CHEMBL2172214 | US9402842, 57)
Affinity DataEC50: >3.47E+4nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50396237(CHEMBL2172208)
Affinity DataEC50:  4.22E+3nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427897(CHEMBL2324622)
Affinity DataEC50:  1.00E+4nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427898(CHEMBL242857)
Affinity DataEC50:  4.84E+3nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50032671(6-[1-(3,5,5,8,8-PENTAMETHYL-5,6,7,8-TETRAHYDRONAPH...)
Affinity DataEC50:  40nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427891(CHEMBL2323836)
Affinity DataEC50:  1.95E+4nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50425046(CHEMBL2312571 | US9402842, 23)
Affinity DataEC50: >4.45E+4nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed