Compile Data Set for Download or QSAR
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Found 32 Enz. Inhib. hit(s) with all data for entry = 50042869
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430432(CHEMBL2334705)
Affinity DataIC50:  1.09E+3nMAssay Description:Inhibition of JNK3 in human SH-SY5Y cells assessed as decrease in anisomycin-induced TNFalpha mRNA level incubated for 1 hr prior to anisomycin induc...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50432394(CHEMBL2348581)
Affinity DataIC50:  1.86E+3nMAssay Description:Competitive inhibition of JNK3 (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50432394(CHEMBL2348581)
Affinity DataIC50:  2.18E+3nMAssay Description:Competitive inhibition of JNK2 (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM16018(14,15-diazatetracyclo[7.6.1.0^{2,7}.0^{13,16}]hexa...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of JNK3 in human PBMCs assessed as decrease in LPS-induced TNFalpha mRNA level after 4 hrs by real-time reverse transcription-PCR analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430438(CHEMBL2335068)
Affinity DataKd:  7.69E+3nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430439(CHEMBL2335067)
Affinity DataKd:  1.17E+3nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430440(CHEMBL2335066)
Affinity DataKd:  2.91E+3nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430441(CHEMBL2335065)
Affinity DataKd:  1.93E+3nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430442(CHEMBL2335064)
Affinity DataKd:  2.98E+3nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430443(CHEMBL2334723)
Affinity DataKd:  2.18E+4nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430444(CHEMBL2334722)
Affinity DataKd:  1.77E+3nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430445(CHEMBL2334721)
Affinity DataKd:  743nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430446(CHEMBL2334720)
Affinity DataKd:  2.33E+3nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430447(CHEMBL2334719)
Affinity DataKd:  1.75E+3nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430448(CHEMBL2334718)
Affinity DataKd:  1.38E+4nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430449(CHEMBL2334717)
Affinity DataKd:  1.91E+4nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430450(CHEMBL2334716)
Affinity DataKd:  2.64E+3nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430451(CHEMBL2334715)
Affinity DataKd:  2.77E+4nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430452(CHEMBL2334714)
Affinity DataKd:  6.05E+3nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430453(CHEMBL2334713)
Affinity DataKd:  1.00E+4nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430454(CHEMBL2334712)
Affinity DataKd:  2.45E+4nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430455(CHEMBL2334711)
Affinity DataKd:  1.07E+4nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50432395(CHEMBL2348778)
Affinity DataKd:  1.81E+4nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430458(CHEMBL2334708)
Affinity DataKd:  1.27E+4nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430459(CHEMBL2334707)
Affinity DataKd:  4.65E+3nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430460(CHEMBL2334706)
Affinity DataKd:  5.26E+3nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430432(CHEMBL2334705)
Affinity DataKd:  46nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430437(CHEMBL2335069)
Affinity DataKd:  1.89E+3nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430436(CHEMBL2335070)
Affinity DataKd:  3.17E+4nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430435(CHEMBL2334702)
Affinity DataKd:  1.66E+3nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430433(CHEMBL2334704)
Affinity DataKd:  2.65E+3nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430434(CHEMBL2334703)
Affinity DataKd:  6.00E+3nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed