Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 5772
TargetHexokinase-4(Human)
University of Dundee

LigandPNGBDBM93225(Kinase inhibitor, A2)
Affinity DataIC50: 4.00E+3nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetHexokinase-4(Human)
University of Dundee

LigandPNGBDBM93226(Kinase inhibitor, B1)
Affinity DataIC50: 6.00E+3nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
University of Dundee

LigandPNGBDBM93226(Kinase inhibitor, B1)
Affinity DataIC50: 1.10E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
University of Dundee

LigandPNGBDBM93229(Kinase inhibitor, F3)
Affinity DataIC50: 1.40E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk2(Human)
University of Dundee

LigandPNGBDBM93226(Kinase inhibitor, B1)
Affinity DataIC50: 1.70E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Dundee

LigandPNGBDBM93224(Kinase inhibitor, A1)
Affinity DataIC50: 1.80E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Chicken)
University of Dundee

LigandPNGBDBM93226(Kinase inhibitor, B1)
Affinity DataIC50: 2.00E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-4(Human)
University of Dundee

LigandPNGBDBM93226(Kinase inhibitor, B1)
Affinity DataIC50: 2.00E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase Yes(Human)
University of Dundee

LigandPNGBDBM93226(Kinase inhibitor, B1)
Affinity DataIC50: 2.10E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 3(Human)
University of Dundee

LigandPNGBDBM93224(Kinase inhibitor, A1)
Affinity DataIC50: 2.10E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Dundee

LigandPNGBDBM93229(Kinase inhibitor, F3)
Affinity DataIC50: 2.20E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
University of Dundee

LigandPNGBDBM93225(Kinase inhibitor, A2)
Affinity DataIC50: 2.40E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Dundee

LigandPNGBDBM93227(Kinase inhibitor, C2)
Affinity DataIC50: 2.50E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK2(Human)
University of Dundee

LigandPNGBDBM93225(Kinase inhibitor, A2)
Affinity DataIC50: 2.50E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetInsulin-like growth factor 1 receptor(Human)
University of Dundee

LigandPNGBDBM93226(Kinase inhibitor, B1)
Affinity DataIC50: 2.50E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Dundee

LigandPNGBDBM93225(Kinase inhibitor, A2)
Affinity DataIC50: 2.60E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
University of Dundee

LigandPNGBDBM93226(Kinase inhibitor, B1)
Affinity DataIC50: 3.90E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetInsulin-like growth factor 1 receptor(Human)
University of Dundee

LigandPNGBDBM93225(Kinase inhibitor, A2)
Affinity DataIC50: 4.70E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Chicken)
University of Dundee

LigandPNGBDBM93224(Kinase inhibitor, A1)
Affinity DataIC50: 9.70E+4nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Sgk1(Human)
University of Dundee

LigandPNGBDBM93227(Kinase inhibitor, C2)
Affinity DataIC50: 1.10E+5nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetSRSF protein kinase 1(Human)
University of Dundee

LigandPNGBDBM93224(Kinase inhibitor, A1)
Affinity DataIC50: 1.14E+5nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Dundee

LigandPNGBDBM93225(Kinase inhibitor, A2)
Affinity DataIC50: 1.31E+5nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetEphrin type-B receptor 3(Human)
University of Dundee

LigandPNGBDBM93228(Kinase inhibitor, D1)
Affinity DataIC50: 1.58E+5nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
University of Dundee

LigandPNGBDBM93225(Kinase inhibitor, A2)
Affinity DataIC50: 1.88E+5nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
University of Dundee

LigandPNGBDBM93224(Kinase inhibitor, A1)
Affinity DataIC50: 1.96E+5nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 1(Human)
University of Dundee

LigandPNGBDBM93225(Kinase inhibitor, A2)
Affinity DataIC50: 2.52E+5nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 1(Human)
University of Dundee

LigandPNGBDBM93228(Kinase inhibitor, D1)
Affinity DataIC50: 4.69E+5nMAssay Description:Selected compounds were screened against a panel of mammalian kinases. Compounds were supplied in DMSO and screened in duplicates at 100 uM concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2013
Entry Details Article
PubMed