Compile Data Set for Download or QSAR
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Found 10 Enz. Inhib. hit(s) with all data for entry = 50042917
TargetHistamine H3 receptor(Mus musculus)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50352090(CHEMBL1824241)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]-iodoproxyfan from histamine H3 receptor in mouse brain cortex after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Mus musculus)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433200(CHEMBL2375594)
Affinity DataKi:  2.5nMAssay Description:Displacement of [125I]-iodoproxyfan from histamine H3 receptor in mouse brain cortex after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Mus musculus)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433199(CHEMBL2375595)
Affinity DataKi:  4.30nMAssay Description:Displacement of [125I]-iodoproxyfan from histamine H3 receptor in mouse brain cortex after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Mus musculus)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433198(CHEMBL2375588)
Affinity DataKi:  6.30nMAssay Description:Displacement of [125I]-iodoproxyfan from histamine H3 receptor in mouse brain cortex after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Mus musculus)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433194(CHEMBL2375587)
Affinity DataKi:  6.90nMAssay Description:Displacement of [125I]-iodoproxyfan from histamine H3 receptor in mouse brain cortex after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Mus musculus)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433197(CHEMBL2375597)
Affinity DataKi:  7.60nMAssay Description:Displacement of [125I]-iodoproxyfan from histamine H3 receptor in mouse brain cortex after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Mus musculus)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433196(CHEMBL2375593)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]-iodoproxyfan from histamine H3 receptor in mouse brain cortex after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Mus musculus)
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433195(CHEMBL2375591)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]-iodoproxyfan from histamine H3 receptor in mouse brain cortex after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433194(CHEMBL2375587)
Affinity DataIC50:  4.03E+4nMAssay Description:Inhibition of human recombinant CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Bioprojet-Biotech

Curated by ChEMBL
LigandPNGBDBM50433194(CHEMBL2375587)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed