Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50042945
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50433574(CHEMBL2381694)
Affinity DataEC50:  0.224nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptor assessed as effect on acetylcholine-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50433574(CHEMBL2381694)
Affinity DataEC50:  0.225nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptor assessed as effect on acetylcholine-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  0.263nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptor assessed as effect on acetylcholine-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  0.263nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptor assessed as effect on acetylcholine-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  4.60nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  4.60nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50433574(CHEMBL2381694)
Affinity DataEC50:  4.60nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50433574(CHEMBL2381694)
Affinity DataEC50:  4.60nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50433574(CHEMBL2381694)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulation of rat muscarinic M4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed