Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50042952
TargetPlatelet-activating factor acetylhydrolase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50125265(N-(2-Diethylamino-ethyl)-2-[2-(4-fluoro-benzylsulf...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of recombinant human Lp-PLA2 using [3H]PAF as substrate at 10 nM incubated for 5 mins prior to substrate addition measured after 10 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50433667(CHEMBL2380965)
Affinity DataIC50: 0.140nMAssay Description:Inhibition of recombinant human Lp-PLA2 using [3H]PAF as substrate at 10 nM incubated for 5 mins prior to substrate addition measured after 10 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50433665(CHEMBL2380967)
Affinity DataIC50: 0.230nMAssay Description:Inhibition of recombinant human Lp-PLA2 using [3H]PAF as substrate at 10 nM incubated for 5 mins prior to substrate addition measured after 10 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50433661(CHEMBL2380954)
Affinity DataIC50: 0.240nMAssay Description:Inhibition of recombinant human Lp-PLA2 using [3H]PAF as substrate at 10 nM incubated for 5 mins prior to substrate addition measured after 10 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50433658(CHEMBL2380957)
Affinity DataIC50: 0.460nMAssay Description:Inhibition of recombinant human Lp-PLA2 using [3H]PAF as substrate at 10 nM incubated for 5 mins prior to substrate addition measured after 10 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50433664(CHEMBL2380968)
Affinity DataIC50: 0.550nMAssay Description:Inhibition of recombinant human Lp-PLA2 using [3H]PAF as substrate at 10 nM incubated for 5 mins prior to substrate addition measured after 10 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50433666(CHEMBL2380966)
Affinity DataIC50: 0.670nMAssay Description:Inhibition of recombinant human Lp-PLA2 using [3H]PAF as substrate at 10 nM incubated for 5 mins prior to substrate addition measured after 10 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50433660(CHEMBL2380955)
Affinity DataIC50: 0.810nMAssay Description:Inhibition of recombinant human Lp-PLA2 using [3H]PAF as substrate at 10 nM incubated for 5 mins prior to substrate addition measured after 10 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50433656(CHEMBL2380959)
Affinity DataIC50: 0.860nMAssay Description:Inhibition of recombinant human Lp-PLA2 using [3H]PAF as substrate at 10 nM incubated for 5 mins prior to substrate addition measured after 10 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50433659(CHEMBL2380956)
Affinity DataIC50: 0.890nMAssay Description:Inhibition of recombinant human Lp-PLA2 using [3H]PAF as substrate at 10 nM incubated for 5 mins prior to substrate addition measured after 10 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50433668(CHEMBL2380963)
Affinity DataIC50: 0.910nMAssay Description:Inhibition of recombinant human Lp-PLA2 using [3H]PAF as substrate at 10 nM incubated for 5 mins prior to substrate addition measured after 10 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50433655(CHEMBL2380960)
Affinity DataIC50: 0.950nMAssay Description:Inhibition of recombinant human Lp-PLA2 using [3H]PAF as substrate at 10 nM incubated for 5 mins prior to substrate addition measured after 10 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50433657(CHEMBL2380958)
Affinity DataIC50: 0.960nMAssay Description:Inhibition of recombinant human Lp-PLA2 using [3H]PAF as substrate at 10 nM incubated for 5 mins prior to substrate addition measured after 10 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50433663(CHEMBL2380859)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of recombinant human Lp-PLA2 using [3H]PAF as substrate at 10 nM incubated for 5 mins prior to substrate addition measured after 10 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50433662(CHEMBL2380952)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of recombinant human Lp-PLA2 using [3H]PAF as substrate at 10 nM incubated for 5 mins prior to substrate addition measured after 10 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed