Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50042882
TargetAdenosine receptor A3(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50420419(CHEMBL2089337)
Affinity DataKi:  13nMAssay Description:Partial agonist activity at human A3 adenosine receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50420427(CHEMBL2089346)
Affinity DataKi:  20nMAssay Description:Antagonist activity at A3 adenosine receptor (unknown origin) assessed as inhibition of adenylate cyclase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50432633(CHEMBL2347371)
Affinity DataKi:  40nMAssay Description:Displacement of [125I]I-AB-MECA from human recombinant A3 adenosine receptor transfected in CHO cells after 60 mins by liquid scintillation counting ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50432634(CHEMBL2347374)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]DPCPX from human recombinant A1 adenosine receptor transfected in CHO cells after 60 mins by liquid scintillation counting analys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50432634(CHEMBL2347374)
Affinity DataKi:  740nMAssay Description:Displacement of [3H]CGS21680 from human A2A adenosine receptor transfected in HEK293 cells after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed