Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50043104
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50436116(CHEMBL2397452)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]-methyl-alpha-D-glucopyranoside accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50436115(CHEMBL2397450)
Affinity DataIC50: 8.90nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]-methyl-alpha-D-glucopyranoside accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50436114(CHEMBL2397451)
Affinity DataIC50: 14nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]-methyl-alpha-D-glucopyranoside accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50436113(CHEMBL2397449)
Affinity DataIC50: 16nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]-methyl-alpha-D-glucopyranoside accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50436112(CHEMBL2397453)
Affinity DataIC50: 17nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]-methyl-alpha-D-glucopyranoside accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50436111(CHEMBL2397442)
Affinity DataIC50: 22nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]-methyl-alpha-D-glucopyranoside accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50436110(CHEMBL2397447)
Affinity DataIC50: 39nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]-methyl-alpha-D-glucopyranoside accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50436109(CHEMBL2397448)
Affinity DataIC50: 70nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]-methyl-alpha-D-glucopyranoside accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50436108(CHEMBL2397441)
Affinity DataIC50: 99nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]-methyl-alpha-D-glucopyranoside accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50436120(CHEMBL2397445)
Affinity DataIC50: 970nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]-methyl-alpha-D-glucopyranoside accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50436119(CHEMBL2397444)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]-methyl-alpha-D-glucopyranoside accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50436118(CHEMBL2397446)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]-methyl-alpha-D-glucopyranoside accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Astellas Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50436117(CHEMBL2397443)
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells assessed as [14C]-methyl-alpha-D-glucopyranoside accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed