Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50005336
TargetDelta-type opioid receptor(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50001683(CHEMBL294616 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataEC50:  6.30nMAssay Description:Agonist activity at human delta opioid receptor transfected in CHOK1 cells after 60 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50491190(CHEMBL2375656)
Affinity DataEC50:  239nMAssay Description:Agonist activity at human delta opioid receptor transfected in CHOK1 cells after 60 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50491190(CHEMBL2375656)
Affinity DataKi:  7.31E+3nMAssay Description:Displacement of [3H]-enkephalin from human delta opioid receptor transfected in CHOK1 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50491190(CHEMBL2375656)
Affinity DataIC50: 1.46E+4nMAssay Description:Displacement of [3H]-enkephalin from human delta opioid receptor transfected in CHOK1 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed