Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50043368
TargetG-protein coupled estrogen receptor 1(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at GPR30 (unknown origin) by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetG-protein coupled estrogen receptor 1(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50303803(cid_5322399 | cid_3136849 | CHEMBL569766 | 1-((3aS...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at GPR30 (unknown origin) by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetG-protein coupled estrogen receptor 1(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of estrogen binding to GPR30 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetG-protein coupled estrogen receptor 1(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50303803(cid_5322399 | cid_3136849 | CHEMBL569766 | 1-((3aS...)
Affinity DataKi:  11nMAssay Description:Inhibition of estrogen binding to GPR30 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed