Affinity DataEC50: 103nMAssay Description:Agonist activity at human LXRbeta-LBD assessed as recruitment of co-activator peptide after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.25E+5nMAssay Description:Agonist activity at human LXRbeta-LBD assessed as recruitment of co-activator peptide after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at human LXRalpha-LBD assessed as recruitment of co-activator peptide after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 91nMAssay Description:Agonist activity at human LXRalpha-LBD assessed as recruitment of co-activator peptide after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKd: 2.20E+3nMAssay Description:Binding affinity to human LXRalpha-LBD by surface plasmon resonanceMore data for this Ligand-Target Pair
Affinity DataKd: 103nMAssay Description:Binding affinity to human LXRbeta-LBD by surface plasmon resonanceMore data for this Ligand-Target Pair
Affinity DataKd: 7.32E+4nMAssay Description:Binding affinity to human LXRbeta-LBD by surface plasmon resonanceMore data for this Ligand-Target Pair
Affinity DataKd: 92nMAssay Description:Binding affinity to human LXRalpha-LBD by surface plasmon resonanceMore data for this Ligand-Target Pair
Affinity DataEC50: 3.50E+3nMAssay Description:Agonist activity at human LXRalpha-LBD assessed as recruitment of co-activator peptide after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair