Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50043334
TargetCyclin-dependent kinase 5 activator 1(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50059889(3-methoxy-2-methyl-4-methylamino-(2S,3S,4S,6R)-29-...)
Affinity DataIC50: 100nMAssay Description:Inhibition of CDK5/p25 (unknown origin)-mediated incorporation of gamma33P into substrate after 20 mins by scintillation counting analysis in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM7262(NSC 705701 | BDBM84528 | alsterpaullone | 9-Nitrop...)
Affinity DataIC50: 330nMAssay Description:Inhibition of CDK5/p25 (unknown origin) after 30 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 930nMAssay Description:Inhibition of CDK5/p25 (unknown origin) after 30 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50439491(AUREUSIDIN)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of CDK5/p25 (unknown origin) after 30 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50439491(AUREUSIDIN)
Affinity DataIC50: 4.81E+3nMAssay Description:Inhibition of CDK5/p25 (unknown origin)-mediated incorporation of gamma33P into substrate after 20 mins by scintillation counting analysis in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50323213(cupressuflavone | CHEMBL1208973)
Affinity DataIC50: 9.29E+3nMAssay Description:Inhibition of CDK5/p25 (unknown origin) after 30 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50241354(Quercetin 3-O-beta-D-glucoside | quercetin 3-O-glu...)
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of CDK5/p25 (unknown origin) after 30 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50439490(CHEMBL2417912)
Affinity DataIC50: 2.23E+4nMAssay Description:Inhibition of CDK5/p25 (unknown origin) after 30 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50439490(CHEMBL2417912)
Affinity DataIC50: 2.43E+4nMAssay Description:Inhibition of CDK5/p25 (unknown origin)-mediated incorporation of gamma33P into substrate after 20 mins by scintillation counting analysis in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50580(MLS000863576 | (2Z)-2-[(3,4-dihydroxyphenyl)methyl...)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of CDK5/p25 (unknown origin) after 30 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50439489(CHEMBL2417913)
Affinity DataIC50: 4.44E+4nMAssay Description:Inhibition of CDK5/p25 (unknown origin) after 30 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50439489(CHEMBL2417913)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CDK5/p25 (unknown origin)-mediated incorporation of gamma33P into substrate after 20 mins by scintillation counting analysis in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed