Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50005719
TargetDNA topoisomerase 2-alpha(Human)
University of Genoa

Curated by ChEMBL
LigandPNGBDBM50493837(CHEMBL2443298)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
University of Genoa

Curated by ChEMBL
LigandPNGBDBM50493837(CHEMBL2443298)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
University of Genoa

Curated by ChEMBL
LigandPNGBDBM50493846(CHEMBL2443290)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
University of Genoa

Curated by ChEMBL
LigandPNGBDBM50493838(CHEMBL2443297)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
University of Genoa

Curated by ChEMBL
LigandPNGBDBM50493835(CHEMBL2443288)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
University of Genoa

Curated by ChEMBL
LigandPNGBDBM50493842(CHEMBL2443291)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
University of Genoa

Curated by ChEMBL
LigandPNGBDBM241949(US9428466, Merbarone)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
University of Genoa

Curated by ChEMBL
LigandPNGBDBM50493841(CHEMBL2443289)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
University of Genoa

Curated by ChEMBL
LigandPNGBDBM50493845(CHEMBL2443300)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
University of Genoa

Curated by ChEMBL
LigandPNGBDBM50493844(CHEMBL2440361)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
University of Genoa

Curated by ChEMBL
LigandPNGBDBM50493843(CHEMBL2443296)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
University of Genoa

Curated by ChEMBL
LigandPNGBDBM50493839(CHEMBL2443292)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
University of Genoa

Curated by ChEMBL
LigandPNGBDBM50493840(CHEMBL2440360)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDNA topoisomerase 2-alpha(Human)
University of Genoa

Curated by ChEMBL
LigandPNGBDBM50493836(CHEMBL2443299)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human topoisomerase 2alpha-mediated relaxation of supercoiled pBR322 after 1 hr by ethidium bromide stainingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed