Compile Data Set for Download or QSAR
maximum 50k data
Found 24 Enz. Inhib. hit(s) with all data for entry = 50005692
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50493693(CHEMBL2434973)
Affinity DataEC50:  347nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50323689(3-amino-N-(4-fluorobenzyl)-4,6-dimethylthieno[2,3-...)
Affinity DataEC50:  219nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM48056(3-amino-N-(2,3-difluorobenzyl)-4,6-dimethyl-thieno...)
Affinity DataEC50:  105nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM48045(3-amino-N-(2-fluorobenzyl)-4,6-dimethyl-thieno[2,3...)
Affinity DataEC50:  126nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM48043(3-amino-4,6-dimethyl-N-p-anisyl-thieno[2,3-b]pyrid...)
Affinity DataEC50:  129nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50493694(CHEMBL2435361)
Affinity DataEC50:  100nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM48054(3-amino-N-(2,5-difluorobenzyl)-4,6-dimethyl-thieno...)
Affinity DataEC50:  130nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50323689(3-amino-N-(4-fluorobenzyl)-4,6-dimethylthieno[2,3-...)
Affinity DataEC50:  220nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50493695(CHEMBL2435355)
Affinity DataEC50:  310nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM48043(3-amino-4,6-dimethyl-N-p-anisyl-thieno[2,3-b]pyrid...)
Affinity DataEC50:  130nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50493696(CHEMBL2435359)
Affinity DataEC50:  580nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50493697(CHEMBL2435349)
Affinity DataEC50:  562nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50493698(CHEMBL2435362)
Affinity DataEC50:  240nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50493698(CHEMBL2435362)
Affinity DataEC50:  240nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM48054(3-amino-N-(2,5-difluorobenzyl)-4,6-dimethyl-thieno...)
Affinity DataEC50:  132nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50493699(CHEMBL2435360)
Affinity DataEC50:  141nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50493695(CHEMBL2435355)
Affinity DataEC50:  309nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50493693(CHEMBL2434973)
Affinity DataEC50:  350nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM48056(3-amino-N-(2,3-difluorobenzyl)-4,6-dimethyl-thieno...)
Affinity DataEC50:  110nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM48045(3-amino-N-(2-fluorobenzyl)-4,6-dimethyl-thieno[2,3...)
Affinity DataEC50:  130nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50493696(CHEMBL2435359)
Affinity DataEC50:  575nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50493697(CHEMBL2435349)
Affinity DataEC50:  560nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50493699(CHEMBL2435360)
Affinity DataEC50:  140nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50493694(CHEMBL2435361)
Affinity DataEC50:  100nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed