Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50005693
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50030474(Avandamet | Avandaryl | Avandia | BRL-49653 | CHEB...)
Affinity DataIC50:  159nMAssay Description:Displacement of fluormone from human PPARgamma LBD expressed in Escherichia coli BL21 DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM53804(4-({2-[(1,3-dioxo-1,3-dihydro-2H-inden-2-ylidene)m...)
Affinity DataIC50:  1.14E+3nMAssay Description:Displacement of fluormone from human PPARgamma LBD expressed in Escherichia coli BL21 DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50387185(CHEMBL2048021)
Affinity DataIC50:  2.22E+3nMAssay Description:Displacement of fluormone from human PPARgamma LBD expressed in Escherichia coli BL21 DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50493700(CHEMBL1426715)
Affinity DataIC50:  5.13E+3nMAssay Description:Displacement of fluormone from human PPARgamma LBD expressed in Escherichia coli BL21 DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed