Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50043542
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442739BDBM50442739(CHEMBL2442801)
Affinity DataIC50: 9.60nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442740BDBM50442740(CHEMBL2442800)
Affinity DataIC50: 49nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442737BDBM50442737(CHEMBL2442691)
Affinity DataIC50: 53nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442721BDBM50442721(CHEMBL2442797)
Affinity DataIC50: 69nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442736BDBM50442736(CHEMBL2442692)
Affinity DataIC50: 69nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442720BDBM50442720(CHEMBL2442798)
Affinity DataIC50: 81nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 19149BDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442723BDBM50442723(CHEMBL2442795)
Affinity DataIC50: 111nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442728BDBM50442728(CHEMBL2442790)
Affinity DataIC50: 130nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442738BDBM50442738(CHEMBL2442802)
Affinity DataIC50: 155nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442719BDBM50442719(CHEMBL2442799)
Affinity DataIC50: 188nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442727BDBM50442727(CHEMBL2442791)
Affinity DataIC50: 193nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442735BDBM50442735(CHEMBL2442693)
Affinity DataIC50: 217nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442731BDBM50442731(CHEMBL2442698)
Affinity DataIC50: 230nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442724BDBM50442724(CHEMBL2442794)
Affinity DataIC50: 242nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442732BDBM50442732(CHEMBL2442697)
Affinity DataIC50: 520nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442729BDBM50442729(CHEMBL2442789)
Affinity DataIC50: 590nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442726BDBM50442726(CHEMBL2442792)
Affinity DataIC50: 767nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442722BDBM50442722(CHEMBL2442796)
Affinity DataIC50: 899nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442725BDBM50442725(CHEMBL2442793)
Affinity DataIC50: 1.44E+3nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 24624BDBM24624(MGCD-0103 | N-(2-aminophenyl)-4-({[4-(pyridin-3-yl...)
Affinity DataIC50: 1.67E+3nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442733BDBM50442733(CHEMBL2442696)
Affinity DataIC50: 1.69E+3nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442730BDBM50442730(CHEMBL2442699)
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442734BDBM50442734(CHEMBL2442694)
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus infected insect high5 cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed