Compile Data Set for Download or QSAR
Report error Found 96 Enz. Inhib. hit(s) with all data for entry = 50044154
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50241748BDBM50241748(dihydro-beta-erythroidine | CHEMBL518059)
Affinity DataKi:  98nMAssay Description:Displacement of [3H]cytisine from alpha4/beta2 nAChR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006634BDBM50006634(CHEMBL3235510)
Affinity DataKi:  550nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006632BDBM50006632(CHEMBL3235508)
Affinity DataIC50: 580nMAssay Description:Antagonist activity at mouse alpha4/beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006648BDBM50006648(CHEBI:4838 | ERYSOTRINE)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]cytisine from alpha4/beta2 nAChR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50014648BDBM50014648(CHEMBL555787 | 6,7-Dimethoxy-2-methyl-1,2,3,4-tetr...)
Affinity DataKi:  870nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006632BDBM50006632(CHEMBL3235508)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006640BDBM50006640(CHEMBL593001)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006638BDBM50006638(CHEMBL2140445)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006630BDBM50006630(CHEMBL3235506)
Affinity DataIC50: 2.30E+3nMAssay Description:Antagonist activity at mouse alpha4/beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006638BDBM50006638(CHEMBL2140445)
Affinity DataIC50: 2.60E+3nMAssay Description:Antagonist activity at mouse alpha4/beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006631BDBM50006631(CHEMBL3235507)
Affinity DataIC50: 2.90E+3nMAssay Description:Antagonist activity at mouse alpha4/beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006634BDBM50006634(CHEMBL3235510)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at mouse alpha4/beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006636BDBM50006636(CHEMBL3235512)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006640BDBM50006640(CHEMBL593001)
Affinity DataIC50: 4.40E+3nMAssay Description:Antagonist activity at mouse alpha4/beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006633BDBM50006633(CHEMBL3235509)
Affinity DataKi:  5.50E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50014647BDBM50014647(CHEMBL544714 | 1,2-Dimethyl-1,2,3,4-tetrahydro-iso...)
Affinity DataKi:  6.80E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006629BDBM50006629(CHEMBL3235505)
Affinity DataKi:  7.30E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006647BDBM50006647(Erysodine)
Affinity DataKi:  7.50E+3nMAssay Description:Displacement of [3H]cytisine from alpha7 nAChR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006630BDBM50006630(CHEMBL3235506)
Affinity DataKi:  8.50E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006629BDBM50006629(CHEMBL3235505)
Affinity DataIC50: 9.20E+3nMAssay Description:Antagonist activity at mouse alpha4/beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006639BDBM50006639(CHEMBL3235514)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50241748BDBM50241748(dihydro-beta-erythroidine | CHEMBL518059)
Affinity DataKi:  1.05E+4nMAssay Description:Displacement of [3H]cytisine from alpha7 nAChR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006637BDBM50006637(CHEMBL3235513)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50014648BDBM50014648(CHEMBL555787 | 6,7-Dimethoxy-2-methyl-1,2,3,4-tetr...)
Affinity DataIC50: 1.20E+4nMAssay Description:Antagonist activity at mouse alpha4/beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50014647BDBM50014647(CHEMBL544714 | 1,2-Dimethyl-1,2,3,4-tetrahydro-iso...)
Affinity DataIC50: 1.60E+4nMAssay Description:Antagonist activity at mouse alpha4/beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006631BDBM50006631(CHEMBL3235507)
Affinity DataKi:  1.80E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006632BDBM50006632(CHEMBL3235508)
Affinity DataKi:  1.90E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006634BDBM50006634(CHEMBL3235510)
Affinity DataKi:  2.10E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006631BDBM50006631(CHEMBL3235507)
Affinity DataKi:  2.30E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006636BDBM50006636(CHEMBL3235512)
Affinity DataIC50: 2.30E+4nMAssay Description:Antagonist activity at mouse alpha4/beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50014648BDBM50014648(CHEMBL555787 | 6,7-Dimethoxy-2-methyl-1,2,3,4-tetr...)
Affinity DataKi:  2.70E+4nMAssay Description:Inhibition of MAOA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50014648BDBM50014648(CHEMBL555787 | 6,7-Dimethoxy-2-methyl-1,2,3,4-tetr...)
Affinity DataKi:  2.90E+4nMAssay Description:Inhibition of MAOB (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006631BDBM50006631(CHEMBL3235507)
Affinity DataKi:  3.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha3/beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006632BDBM50006632(CHEMBL3235508)
Affinity DataKi:  3.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha3/beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006642BDBM50006642(CHEMBL2385327)
Affinity DataKi:  3.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006629BDBM50006629(CHEMBL3235505)
Affinity DataKi:  3.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha3/beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006633BDBM50006633(CHEMBL3235509)
Affinity DataIC50: 3.10E+4nMAssay Description:Antagonist activity at mouse alpha4/beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006628BDBM50006628(CHEMBL3235504)
Affinity DataIC50: 3.10E+4nMAssay Description:Antagonist activity at mouse alpha4/beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006639BDBM50006639(CHEMBL3235514)
Affinity DataIC50: 3.30E+4nMAssay Description:Antagonist activity at mouse alpha4/beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006631BDBM50006631(CHEMBL3235507)
Affinity DataIC50: 3.30E+4nMAssay Description:Antagonist activity at rat alpha3/beta4 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50014648BDBM50014648(CHEMBL555787 | 6,7-Dimethoxy-2-methyl-1,2,3,4-tetr...)
Affinity DataKi:  4.67E+4nMAssay Description:Displacement of [3H]-serotonin from human SERT expressed in African green monkey COS7 cells after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006629BDBM50006629(CHEMBL3235505)
Affinity DataKi:  5.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006630BDBM50006630(CHEMBL3235506)
Affinity DataKi:  5.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006628BDBM50006628(CHEMBL3235504)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at rat alpha3/beta4 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006629BDBM50006629(CHEMBL3235505)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at rat alpha3/beta4 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006637BDBM50006637(CHEMBL3235513)
Affinity DataKi:  5.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006638BDBM50006638(CHEMBL2140445)
Affinity DataKi:  5.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha4/beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006630BDBM50006630(CHEMBL3235506)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at rat alpha3/beta4 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-2(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006635BDBM50006635(CHEMBL3235511)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at mouse alpha4/beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006632BDBM50006632(CHEMBL3235508)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at rat alpha3/beta4 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane pot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
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