Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50043669
TargetProteasome subunit beta type-5(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444464(CHEMBL192046)
Affinity DataEC50:  10nMAssay Description:Inhibition of chymotrypsin like activity of 20S proteasome in HEK293 cells after 24 hrs by microscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50398608(MARIZOMIB)
Affinity DataIC50: 22nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome after 1 hr by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444464(CHEMBL192046)
Affinity DataIC50: 23nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome after 1 hr by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444462(CHEMBL3092609)
Affinity DataIC50: 28nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome after 1 hr by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444463(CHEMBL3092608)
Affinity DataIC50: 50nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome after 1 hr by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444463(CHEMBL3092608)
Affinity DataEC50:  90nMAssay Description:Inhibition of chymotrypsin like activity of 20S proteasome in HEK293 cells after 24 hrs by microscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444466(CHEMBL3092611)
Affinity DataIC50: 330nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome after 1 hr by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444461(CHEMBL3092610)
Affinity DataEC50:  332nMAssay Description:Inhibition of chymotrypsin like activity of 20S proteasome in HEK293 cells after 24 hrs by microscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444462(CHEMBL3092609)
Affinity DataEC50:  360nMAssay Description:Inhibition of chymotrypsin like activity of 20S proteasome in HEK293 cells after 24 hrs by microscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444461(CHEMBL3092610)
Affinity DataIC50: 500nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome after 1 hr by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50444465(CHEMBL3092612)
Affinity DataIC50: 500nMAssay Description:Inhibition of chymotrypsin like activity of human 20S proteasome after 1 hr by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed