Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 50043760
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445826BDBM50445826(CHEMBL3105402)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 27566BDBM27566(4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbo...)
Affinity DataIC50: 10nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 27135BDBM27135(2-[(2R)-2-methylpyrrolidin-2-yl]-1H-1,3-benzodiazo...)
Affinity DataIC50: 10nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445864BDBM50445864(CHEMBL3105398)
Affinity DataIC50: 29nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445825BDBM50445825(CHEMBL3105403)
Affinity DataIC50: 30nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50316226BDBM50316226(MK-4827 | (S)-2-(4-(piperidin-3-yl)phenyl)-2H-inda...)
Affinity DataIC50: 30nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445859BDBM50445859(CHEMBL3105407)
Affinity DataIC50: 32nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445853BDBM50445853(CHEMBL1544030)
Affinity DataIC50: 43nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445854BDBM50445854(CHEMBL3105410)
Affinity DataIC50: 50nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445824BDBM50445824(CHEMBL3105405)
Affinity DataIC50: 56nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445827BDBM50445827(CHEMBL3105399)
Affinity DataIC50: 67nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445856BDBM50445856(CHEMBL3102884)
Affinity DataIC50: 87nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445855BDBM50445855(CHEMBL3105409)
Affinity DataIC50: 88nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445863BDBM50445863(CHEMBL3105400)
Affinity DataIC50: 110nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445862BDBM50445862(CHEMBL3105401)
Affinity DataIC50: 130nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445861BDBM50445861(CHEMBL3105404)
Affinity DataIC50: 130nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445845BDBM50445845(CHEMBL3105416)
Affinity DataIC50: 130nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445850BDBM50445850(CHEMBL3105413)
Affinity DataIC50: 190nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445858BDBM50445858(CHEMBL3105408)
Affinity DataIC50: 220nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445826BDBM50445826(CHEMBL3105402)
Affinity DataEC50:  256nMAssay Description:Inhibition of PARP-1-mediated PARylation in H2O2-induced human HeLa cells preincubated for 3 hrs followed by H2O2 addition measured after 5 mins by D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445839BDBM50445839(CHEMBL3105422)
Affinity DataIC50: 260nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445849BDBM50445849(CHEMBL1508664)
Affinity DataIC50: 270nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445836BDBM50445836(CHEMBL3105424)
Affinity DataIC50: 280nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445828BDBM50445828(CHEMBL3105432)
Affinity DataIC50: 280nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445860BDBM50445860(CHEMBL3105406)
Affinity DataIC50: 300nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445841BDBM50445841(CHEMBL3105420)
Affinity DataIC50: 350nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445843BDBM50445843(CHEMBL3105418)
Affinity DataIC50: 410nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445824BDBM50445824(CHEMBL3105405)
Affinity DataEC50:  467nMAssay Description:Inhibition of PARP-1-mediated PARylation in H2O2-induced human HeLa cells preincubated for 3 hrs followed by H2O2 addition measured after 5 mins by D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445846BDBM50445846(CHEMBL3105415)
Affinity DataIC50: 540nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445835BDBM50445835(CHEMBL3105425)
Affinity DataIC50: 600nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445833BDBM50445833(CHEMBL3105427)
Affinity DataIC50: 600nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445838BDBM50445838(CHEMBL552501)
Affinity DataIC50: 690nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445827BDBM50445827(CHEMBL3105399)
Affinity DataEC50:  707nMAssay Description:Inhibition of PARP-1-mediated PARylation in H2O2-induced human HeLa cells preincubated for 3 hrs followed by H2O2 addition measured after 5 mins by D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445844BDBM50445844(CHEMBL3105417)
Affinity DataIC50: 760nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445831BDBM50445831(CHEMBL3105429)
Affinity DataIC50: 820nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445830BDBM50445830(CHEMBL3105430)
Affinity DataIC50: 820nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445825BDBM50445825(CHEMBL3105403)
Affinity DataEC50:  865nMAssay Description:Inhibition of PARP-1-mediated PARylation in H2O2-induced human HeLa cells preincubated for 3 hrs followed by H2O2 addition measured after 5 mins by D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445848BDBM50445848(CHEMBL1726644)
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445829BDBM50445829(CHEMBL3105431)
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445834BDBM50445834(CHEMBL3105426)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445852BDBM50445852(CHEMBL3105411)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445840BDBM50445840(CHEMBL3105421)
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445842BDBM50445842(CHEMBL3105419)
Affinity DataIC50: 1.52E+3nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50396747BDBM50396747(CHEMBL2172241)
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445837BDBM50445837(CHEMBL3105423)
Affinity DataIC50: 1.86E+3nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445832BDBM50445832(CHEMBL3105428)
Affinity DataIC50: 1.96E+3nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445851BDBM50445851(CHEMBL3105412)
Affinity DataIC50: 2.54E+3nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
R&D Sigma-Tau Industrie Farmaceutiche Riunite

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445847BDBM50445847(CHEMBL3105414)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of GST-tagged recombinant human PARP-1 expressed in Escherichia coli after 30 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed