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Found 33 Enz. Inhib. hit(s) with all data for entry = 50006027
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496304(CHEMBL3125712)
Affinity DataKi:  4.90nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496310(CHEMBL3125713)
Affinity DataKi:  6.70nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496311(CHEMBL3125718)
Affinity DataKi:  7.80nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496307(CHEMBL3125717)
Affinity DataKi:  8.60nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496308(CHEMBL3125714)
Affinity DataKi:  9.20nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496311(CHEMBL3125718)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496305(CHEMBL3125716)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496306(CHEMBL3125711)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496309(CHEMBL3125719)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496305(CHEMBL3125716)
Affinity DataKi:  26nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496308(CHEMBL3125714)
Affinity DataKi:  39nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496309(CHEMBL3125719)
Affinity DataKi:  43nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496303(CHEMBL3125715)
Affinity DataKi:  58nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496307(CHEMBL3125717)
Affinity DataKi:  59nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496306(CHEMBL3125711)
Affinity DataKi:  65nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496306(CHEMBL3125711)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]-CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496303(CHEMBL3125715)
Affinity DataKi:  160nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496310(CHEMBL3125713)
Affinity DataKi:  176nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496304(CHEMBL3125712)
Affinity DataKi:  231nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496303(CHEMBL3125715)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]-R-PIA from recombinant human adenosine A1 receptor expressed in CHO cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496303(CHEMBL3125715)
Affinity DataKi:  1.76E+3nMAssay Description:Displacement of [3H]-CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496308(CHEMBL3125714)
Affinity DataKi:  2.17E+3nMAssay Description:Displacement of [3H]-R-PIA from recombinant human adenosine A1 receptor expressed in CHO cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496308(CHEMBL3125714)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [3H]-CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496305(CHEMBL3125716)
Affinity DataKi:  2.53E+3nMAssay Description:Displacement of [3H]-CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496310(CHEMBL3125713)
Affinity DataKi:  2.86E+3nMAssay Description:Displacement of [3H]-CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496307(CHEMBL3125717)
Affinity DataKi:  3.15E+3nMAssay Description:Displacement of [3H]-CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496311(CHEMBL3125718)
Affinity DataKi:  3.31E+3nMAssay Description:Displacement of [3H]-CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496304(CHEMBL3125712)
Affinity DataKi:  7.49E+3nMAssay Description:Displacement of [3H]-CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496304(CHEMBL3125712)
Affinity DataEC50:  46nMAssay Description:Partial agonist activity at recombinant human adenosine A3 receptor expressed in CHO cells assessed as stimulation of forskolin-induced intracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496309(CHEMBL3125719)
Affinity DataEC50:  19nMAssay Description:Partial agonist activity at recombinant human adenosine A3 receptor expressed in CHO cells assessed as stimulation of forskolin-induced intracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496308(CHEMBL3125714)
Affinity DataEC50:  20nMAssay Description:Partial agonist activity at recombinant human adenosine A3 receptor expressed in CHO cells assessed as stimulation of forskolin-induced intracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496310(CHEMBL3125713)
Affinity DataEC50:  16nMAssay Description:Partial agonist activity at recombinant human adenosine A3 receptor expressed in CHO cells assessed as stimulation of forskolin-induced intracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496303(CHEMBL3125715)
Affinity DataEC50:  27nMAssay Description:Partial agonist activity at recombinant human adenosine A3 receptor expressed in CHO cells assessed as stimulation of forskolin-induced intracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed