Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50044325
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013050BDBM50013050(CHEMBL3261693)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013071BDBM50013071(CHEMBL3261688)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013051BDBM50013051(CHEMBL3261694)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013112BDBM50013112(CHEMBL3261704)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013103BDBM50013103(CHEMBL3261692)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013053BDBM50013053(CHEMBL3261696)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013104BDBM50013104(CHEMBL3261697)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013117BDBM50013117(CHEMBL3261691)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 30130BDBM30130(Prozac | cid_62857 | Fluoxetin | CHEMBL41 | CHEMBL...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013079BDBM50013079(CHEMBL3261689)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013069BDBM50013069(CHEMBL3261686)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013056BDBM50013056(CHEMBL3261699)
Affinity DataKi:  9.40nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013065BDBM50013065(CHEMBL3261703)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013102BDBM50013102(CHEMBL3261690)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013070BDBM50013070(CHEMBL3261687)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013052BDBM50013052(CHEMBL3261695)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013054BDBM50013054(CHEMBL3261698)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013067BDBM50013067(CHEMBL3261707)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013069BDBM50013069(CHEMBL3261686)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013070BDBM50013070(CHEMBL3261687)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013068BDBM50013068(CHEMBL3261708)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013057BDBM50013057(CHEMBL3261700)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013054BDBM50013054(CHEMBL3261698)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013066BDBM50013066(CHEMBL3261706)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013102BDBM50013102(CHEMBL3261690)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013052BDBM50013052(CHEMBL3261695)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013066BDBM50013066(CHEMBL3261706)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013058BDBM50013058(CHEMBL3261701)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013050BDBM50013050(CHEMBL3261693)
Affinity DataKi:  61nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013071BDBM50013071(CHEMBL3261688)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013058BDBM50013058(CHEMBL3261701)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013064BDBM50013064(CHEMBL3261702)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013057BDBM50013057(CHEMBL3261700)
Affinity DataKi:  88nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013064BDBM50013064(CHEMBL3261702)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013068BDBM50013068(CHEMBL3261708)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013053BDBM50013053(CHEMBL3261696)
Affinity DataKi:  96nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013065BDBM50013065(CHEMBL3261703)
Affinity DataKi:  102nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 30130BDBM30130(Prozac | cid_62857 | Fluoxetin | CHEMBL41 | CHEMBL...)
Affinity DataKi:  109nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013051BDBM50013051(CHEMBL3261694)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82272BDBM82272(SB 200646 | SB200646a)
Affinity DataKi:  124nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013103BDBM50013103(CHEMBL3261692)
Affinity DataKi:  135nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013067BDBM50013067(CHEMBL3261707)
Affinity DataKi:  152nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013113BDBM50013113(CHEMBL3261705)
Affinity DataKi:  197nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013056BDBM50013056(CHEMBL3261699)
Affinity DataKi:  652nMAssay Description:Displacement of [3H]mesulergine from 5-HT2C receptor in Sprague-Dawley rat choroid plexus membranes after 30 mins by liquid scintillation spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82272BDBM82272(SB 200646 | SB200646a)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013079BDBM50013079(CHEMBL3261689)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat whole brain membranes after 1 hr by liquid scintillation spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed