Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50044147
TargetProlyl endopeptidase(Human)
University of Helsinki

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155838BDBM50155838((S)-1-((S)-1-(4-phenylbutanoyl)pyrrolidine-2-carbo...)
Affinity DataKi:  0.0230nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155838BDBM50155838((S)-1-((S)-1-(4-phenylbutanoyl)pyrrolidine-2-carbo...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of porcine prolyl oligopeptidase using Z-Gly-Pro-AMC as substrate after 60 mins by double-reciprocal plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProlyl endopeptidase(Rat)
University of Helsinki

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005864BDBM50005864(CHEMBL3236270)
Affinity DataKi:  0.950nMAssay Description:Competitive inhibition of rat brain prolyl oligopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProlyl endopeptidase(Human)
University of Helsinki

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50051539BDBM50051539(4-Phenyl-1-[2-(pyrrolidine-1-carbonyl)-pyrrolidin-...)
Affinity DataKi:  0.970nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProlyl endopeptidase(Mouse)
University of Helsinki

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005870BDBM50005870(CHEMBL3236271)
Affinity DataIC50: 3.10nMAssay Description:Competitive inhibition of mouse brain prolyl oligopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005880BDBM50005880(CHEMBL3236273)
Affinity DataKi:  4.20nMAssay Description:Inhibition of porcine prolyl oligopeptidase using Z-Gly-Pro-AMC as substrate after 60 mins by double-reciprocal plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProlyl endopeptidase(Pig)
University of Helsinki

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005872BDBM50005872(CHEMBL3236272)
Affinity DataKi:  22nMAssay Description:Inhibition of porcine prolyl oligopeptidase using Z-Gly-Pro-AMC as substrate after 60 mins by double-reciprocal plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed