Compile Data Set for Download or QSAR
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Found 7 Enz. Inhib. hit(s) with all data for entry = 50044147
TargetProlyl endopeptidase(Homo sapiens (Human))
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50155838((S)-1-((S)-1-(4-phenylbutanoyl)pyrrolidine-2-carbo...)
Affinity DataKi:  0.0230nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
TargetProlyl endopeptidase(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50155838((S)-1-((S)-1-(4-phenylbutanoyl)pyrrolidine-2-carbo...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of porcine prolyl oligopeptidase using Z-Gly-Pro-AMC as substrate after 60 mins by double-reciprocal plot analysisMore data for this Ligand-Target Pair
TargetProlyl endopeptidase(Rattus norvegicus)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50005864(CHEMBL3236270)
Affinity DataKi:  0.950nMAssay Description:Competitive inhibition of rat brain prolyl oligopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50051539((S)-4-phenyl-1-(2-(pyrrolidine-1-carbonyl)pyrrolid...)
Affinity DataKi:  0.970nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50005880(CHEMBL3236273)
Affinity DataKi:  4.20nMAssay Description:Inhibition of porcine prolyl oligopeptidase using Z-Gly-Pro-AMC as substrate after 60 mins by double-reciprocal plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50005872(CHEMBL3236272)
Affinity DataKi:  22nMAssay Description:Inhibition of porcine prolyl oligopeptidase using Z-Gly-Pro-AMC as substrate after 60 mins by double-reciprocal plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Mus musculus)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50005870(CHEMBL3236271)
Affinity DataIC50:  3.10nMAssay Description:Competitive inhibition of mouse brain prolyl oligopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed