Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50044502
TargetMuscarinic acetylcholine receptor M2(Human)
Keio University

Curated by ChEMBL
LigandPNGBDBM50019290(CHEMBL3289390)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]NMS from human M2R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Keio University

Curated by ChEMBL
LigandPNGBDBM50377964(Cantil | Glycophenylate | Mepenzolate | MEPENZOLAT...)
Affinity DataKi:  0.680nMAssay Description:Displacement of [3H]NMS from human M2R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Keio University

Curated by ChEMBL
LigandPNGBDBM50019290(CHEMBL3289390)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]NMS from human M3R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Keio University

Curated by ChEMBL
LigandPNGBDBM50019289(CHEMBL3289391)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]NMS from human M2R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Keio University

Curated by ChEMBL
LigandPNGBDBM50377964(Cantil | Glycophenylate | Mepenzolate | MEPENZOLAT...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]NMS from human M3R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Keio University

Curated by ChEMBL
LigandPNGBDBM50019289(CHEMBL3289391)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]NMS from human M3R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed