Affinity DataKi: 14nMAssay Description:Binding affinity to human alpha7 nAChRMore data for this Ligand-Target Pair
Affinity DataIC50: 5.60E+3nMAssay Description:Competitive antagonist activity at human alpha7 nAChR expressed in Xenopus oocyte assessed as inhibition of ACh-induced current by voltage clamp meth...More data for this Ligand-Target Pair
Affinity DataIC50: 6.10E+3nMAssay Description:Non competitive antagonist activity at human alpha7 nAChR expressed in Xenopus oocyte assessed as inhibition of ACh-induced current by voltage clamp ...More data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in Xenopus oocyte assessed as inhibition of ACh-induced current by voltage clamp methodMore data for this Ligand-Target Pair
Affinity DataIC50: 7.20E+3nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in Xenopus oocyte assessed as inhibition of ACh-induced current by voltage clamp methodMore data for this Ligand-Target Pair
Affinity DataEC50: 6.90E+4nMAssay Description:Agonist activity at human recombinant alpha7 nAChR expressed in Xenopus oocyte in presence of 6 uM (S)-ethyl 1-(2-cyanoethyl)pyrrolidine-2-carboxylat...More data for this Ligand-Target Pair
Affinity DataEC50: 8.70E+4nMAssay Description:Agonist activity at human recombinant alpha7 nAChR expressed in Xenopus oocyteMore data for this Ligand-Target Pair
Affinity DataEC50: 4.40E+3nMAssay Description:Partial agonist activity at human alpha7 nAChR expressed in Xenopus oocyte assessed as evoked ACh-induced current by voltage clamp methodMore data for this Ligand-Target Pair