Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50042590
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428271BDBM50428271(CHEMBL2337032)
Affinity DataKd:  270nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428273BDBM50428273(CHEMBL2337030)
Affinity DataKd:  590nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428274BDBM50428274(CHEMBL2337029)
Affinity DataKd:  630nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428272BDBM50428272(CHEMBL2337031)
Affinity DataKd:  680nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428268BDBM50428268(CHEMBL2337017)
Affinity DataKd:  710nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428239BDBM50428239(CHEMBL2337448)
Affinity DataKd:  1.10E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428238BDBM50428238(CHEMBL2337449)
Affinity DataKd:  1.10E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428236BDBM50428236(CHEMBL1457864)
Affinity DataKd:  1.40E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428267BDBM50428267(CHEMBL2337018)
Affinity DataKd:  1.50E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428240BDBM50428240(CHEMBL2337447)
Affinity DataKd:  1.80E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428256BDBM50428256(CHEMBL2337027)
Affinity DataKd:  2.20E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428235BDBM50428235(CHEMBL2337028)
Affinity DataKd:  3.10E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428257BDBM50428257(CHEMBL2337026)
Affinity DataKd:  3.50E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428252BDBM50428252(CHEMBL2337034)
Affinity DataKd:  4.70E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428270BDBM50428270(CHEMBL1407785)
Affinity DataKd:  5.80E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428255BDBM50428255(CHEMBL1231559)
Affinity DataIC50: 6.00E+3nMAssay Description:Antagonist activity at WDR5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428263BDBM50428263(CHEMBL2337021)
Affinity DataKd:  6.60E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428254BDBM50428254(CHEMBL1609857)
Affinity DataKd:  6.90E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428254BDBM50428254(CHEMBL1609857)
Affinity DataKd:  7.00E+3nMAssay Description:Displacement of MLL-WIN N-terminal FITC-tagged GSARAEVHLRKS peptide from human WDR5 (1-334) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428251BDBM50428251(CHEMBL2337035)
Affinity DataKd:  7.00E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428237BDBM50428237(CHEMBL2337450)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428269BDBM50428269(CHEMBL2337016)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428258BDBM50428258(CHEMBL2337025)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428259BDBM50428259(CHEMBL2331612)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428241BDBM50428241(CHEMBL2337446)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428262BDBM50428262(CHEMBL2337022)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428260BDBM50428260(CHEMBL2337024)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428261BDBM50428261(CHEMBL2337023)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428266BDBM50428266(CHEMBL2337019)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428264BDBM50428264(CHEMBL1559278)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428265BDBM50428265(CHEMBL2337020)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428247BDBM50428247(CHEMBL2337039)
Affinity DataKd:  1.58E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428253BDBM50428253(CHEMBL2337033)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428243BDBM50428243(CHEMBL2337444)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428244BDBM50428244(CHEMBL2337443)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428242BDBM50428242(CHEMBL2337445)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428248BDBM50428248(CHEMBL2337038)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428245BDBM50428245(CHEMBL2337442)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428246BDBM50428246(CHEMBL2337441)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428249BDBM50428249(CHEMBL2337037)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50428250BDBM50428250(CHEMBL2337036)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed