Compile Data Set for Download or QSAR
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Found 6 Enz. Inhib. hit(s) with all data for entry = 50044275
TargetMitotic checkpoint serine/threonine-protein kinase BUB1(Homo sapiens (Human))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011209(CHEMBL3260324)
Affinity DataIC50:  5nMAssay Description:Inhibition of Bub1 kinase (unknown origin) by TR-FRET kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitotic checkpoint serine/threonine-protein kinase BUB1(Homo sapiens (Human))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011201(CHEMBL3260326)
Affinity DataIC50:  6nMAssay Description:Inhibition of Bub1 kinase (unknown origin) by TR-FRET kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitotic checkpoint serine/threonine-protein kinase BUB1(Homo sapiens (Human))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011202(CHEMBL3260325)
Affinity DataIC50:  9nMAssay Description:Inhibition of Bub1 kinase (unknown origin) by TR-FRET kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitotic checkpoint serine/threonine-protein kinase BUB1(Homo sapiens (Human))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011188(CHEMBL3260329)
Affinity DataIC50:  30nMAssay Description:Inhibition of Bub1 kinase (unknown origin) by TR-FRET kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitotic checkpoint serine/threonine-protein kinase BUB1(Homo sapiens (Human))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011200(CHEMBL3260327)
Affinity DataIC50:  500nMAssay Description:Inhibition of Bub1 kinase (unknown origin) by TR-FRET kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitotic checkpoint serine/threonine-protein kinase BUB1(Homo sapiens (Human))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011189(CHEMBL3260328)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Bub1 kinase (unknown origin) by TR-FRET kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed