Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50044276
TargeteIF-2-alpha kinase GCN2(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011233(CHEMBL3260331)
Affinity DataIC50: 300nMAssay Description:Inhibition of GCN2-mediated elF2alpha phosphorylation in human U2OS cells after 2 hrs by immunocytochemistryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargeteIF-2-alpha kinase GCN2(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011233(CHEMBL3260331)
Affinity DataIC50: 300nMAssay Description:Inhibition of GCN2 (unknown origin) using GFP-elF2a as substrate preincubated with substrate for 20 mins measured after 90 mins by Lanthascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargeteIF-2-alpha kinase GCN2(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011234(CHEMBL3260330)
Affinity DataIC50: 300nMAssay Description:Inhibition of GCN2-mediated elF2alpha phosphorylation in human U2OS cells after 2 hrs by immunocytochemistryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargeteIF-2-alpha kinase GCN2(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011234(CHEMBL3260330)
Affinity DataIC50: 300nMAssay Description:Inhibition of GCN2 (unknown origin) using GFP-elF2a as substrate preincubated with substrate for 20 mins measured after 90 mins by Lanthascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargeteIF-2-alpha kinase GCN2(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011232(CHEMBL3260332)
Affinity DataIC50: 300nMAssay Description:Inhibition of GCN2-mediated elF2alpha phosphorylation in human U2OS cells after 2 hrs by immunocytochemistryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargeteIF-2-alpha kinase GCN2(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011232(CHEMBL3260332)
Affinity DataIC50: 300nMAssay Description:Inhibition of GCN2 (unknown origin) using GFP-elF2a as substrate preincubated with substrate for 20 mins measured after 90 mins by Lanthascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargeteIF-2-alpha kinase GCN2(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011235(CHEMBL3260333)
Affinity DataIC50: 300nMAssay Description:Inhibition of GCN2 (unknown origin) using GFP-elF2a as substrate preincubated with substrate for 20 mins measured after 90 mins by Lanthascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargeteIF-2-alpha kinase GCN2(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011235(CHEMBL3260333)
Affinity DataIC50: 300nMAssay Description:Inhibition of GCN2-mediated elF2alpha phosphorylation in human U2OS cells after 2 hrs by immunocytochemistryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed