Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50044559
TargetE3 ubiquitin-protein ligase Mdm2(Human)
Cairo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020725BDBM50020725(CHEMBL3291439)
Affinity DataIC50: 260nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
Cairo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020716BDBM50020716(CHEMBL3286447)
Affinity DataIC50: 360nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
Cairo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020717BDBM50020717(CHEMBL3291433)
Affinity DataIC50: 440nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
Cairo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020724BDBM50020724(CHEMBL3291438)
Affinity DataIC50: 550nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
Cairo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020723BDBM50020723(CHEMBL3291437)
Affinity DataIC50: 570nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
Cairo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020722BDBM50020722(CHEMBL3291436)
Affinity DataIC50: 610nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
Cairo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020721BDBM50020721(CHEMBL3291435)
Affinity DataIC50: 780nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
Cairo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020720BDBM50020720(CHEMBL3291434)
Affinity DataIC50: 810nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
Cairo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020715BDBM50020715(CHEMBL3291222)
Affinity DataIC50: 840nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
Cairo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020726BDBM50020726(CHEMBL3291221)
Affinity DataIC50: 890nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
Cairo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020727BDBM50020727(CHEMBL3291220)
Affinity DataIC50: 910nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
Cairo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020728BDBM50020728(CHEMBL3291219)
Affinity DataIC50: 940nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
Cairo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020729BDBM50020729(CHEMBL3291218)
Affinity DataIC50: 970nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
Cairo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020714BDBM50020714(CHEMBL3291217)
Affinity DataIC50: 990nMAssay Description:Inhibition of GST-tagged HDM2 (unknown origin) expressed in Escherichia coli BL21 cells assessed as p53 activation by measuring inhibition of His-p53...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed