Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50044590
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 280nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50021612(CHEMBL3291228)
Affinity DataIC50: 400nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50021604(CHEMBL3290949)
Affinity DataIC50: 430nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50021607(CHEMBL3291224)
Affinity DataIC50: 730nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50021611(CHEMBL3291227)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50021605(CHEMBL3290950)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50021609(CHEMBL3291226)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50021596(CHEMBL3291232)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50021597(CHEMBL3291233)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50021598(CHEMBL3291234)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50021599(CHEMBL3286445)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50021594(CHEMBL3291230)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50021595(CHEMBL3291231)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50021600(CHEMBL3291235)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50021608(CHEMBL3291225)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50021603(CHEMBL3291236)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50021606(CHEMBL3291223)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-33P]ATP after 30 mins incubation by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed