Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50045235
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50051783(CHEMBL3358450)
Affinity DataKi:  15nMAssay Description:Binding affinity to human ghrelin receptor by receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50051718(CHEMBL3358452)
Affinity DataIC50:  4nMAssay Description:Antagonist activity against human ghrelin receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50051748(CHEMBL3358451)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against human ghrelin receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50051709(CHEMBL3358453)
Affinity DataIC50:  38nMAssay Description:Antagonist activity against human ghrelin receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed