Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50006214
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50497864(CHEMBL3319093)
Affinity DataIC50:  2.45E+3nMAssay Description:Antagonist activity against Myc-tagged RXRalpha ligand binding domain (unknown origin) expressed in human HEK293T cells assessed as inhibition of 9-c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50497864(CHEMBL3319093)
Affinity DataKd:  488nMAssay Description:Binding affinity to RXRalpha ligand binding domain (unknown origin) expressed in human HEK293T cells by SPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed