Compile Data Set for Download or QSAR
maximum 50k data
Found 33 Enz. Inhib. hit(s) with all data for entry = 50045291
TargetHistone deacetylase 1(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055512(CHEMBL3317812)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055513(CHEMBL3317811)
Affinity DataIC50:  0.210nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055514(CHEMBL3317810)
Affinity DataIC50:  0.290nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055513(CHEMBL3317811)
Affinity DataIC50:  0.380nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50020912(Largazole Thiol)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055515(CHEMBL3317818)
Affinity DataIC50:  0.620nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055514(CHEMBL3317810)
Affinity DataIC50:  0.680nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50020912(Largazole Thiol)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50020912(Largazole Thiol)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055516(CHEMBL3317817)
Affinity DataIC50:  0.960nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055513(CHEMBL3317811)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055515(CHEMBL3317818)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055515(CHEMBL3317818)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055512(CHEMBL3317812)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055512(CHEMBL3317812)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055516(CHEMBL3317817)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055514(CHEMBL3317810)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055516(CHEMBL3317817)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055517(CHEMBL3317816)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055517(CHEMBL3317816)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055518(CHEMBL3317815)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055517(CHEMBL3317816)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055510(CHEMBL3317814)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055518(CHEMBL3317815)
Affinity DataIC50:  6nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055518(CHEMBL3317815)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055510(CHEMBL3317814)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055510(CHEMBL3317814)
Affinity DataIC50:  21nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055511(CHEMBL3317813)
Affinity DataIC50:  39nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055511(CHEMBL3317813)
Affinity DataIC50:  100nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50020912(Largazole Thiol)
Affinity DataIC50:  102nMAssay Description:Inhibition of HDAC8 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055511(CHEMBL3317813)
Affinity DataIC50:  150nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055515(CHEMBL3317818)
Affinity DataIC50:  540nMAssay Description:Inhibition of HDAC8 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Duke University

Curated by ChEMBL
LigandPNGBDBM50055516(CHEMBL3317817)
Affinity DataIC50:  790nMAssay Description:Inhibition of HDAC8 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed