Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50045303
TargetSerine/threonine-protein kinase pim-3(Human)
Clermont Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055958BDBM50055958(CHEMBL3326555)
Affinity DataIC50: 20nMAssay Description:Inhibition of full-length human PIM3 using RSRHSSYPAGT as substrate assessed as residual kinase activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Clermont Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055958BDBM50055958(CHEMBL3326555)
Affinity DataIC50: 70nMAssay Description:Inhibition of full-length human PIM1 using RSRHSSYPAGT as substrate assessed as residual kinase activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Clermont Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055959BDBM50055959(CHEMBL3326556)
Affinity DataIC50: 120nMAssay Description:Inhibition of full-length human PIM1 using RSRHSSYPAGT as substrate assessed as residual kinase activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Clermont Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055959BDBM50055959(CHEMBL3326556)
Affinity DataIC50: 140nMAssay Description:Inhibition of full-length human PIM3 using RSRHSSYPAGT as substrate assessed as residual kinase activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Clermont Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055961BDBM50055961(CHEMBL3326558)
Affinity DataIC50: 169nMAssay Description:Inhibition of full-length human PIM3 using RSRHSSYPAGT as substrate assessed as residual kinase activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Clermont Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055960BDBM50055960(CHEMBL3326557)
Affinity DataIC50: 200nMAssay Description:Inhibition of full-length human PIM3 using RSRHSSYPAGT as substrate assessed as residual kinase activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Clermont Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055962BDBM50055962(CHEMBL3326559)
Affinity DataIC50: 400nMAssay Description:Inhibition of full-length human PIM3 using RSRHSSYPAGT as substrate assessed as residual kinase activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed