Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50045339
TargetGlucagon receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50122102(3-Cyano-4-hydroxy-benzoic acid [1-(2,3,5,6-tetrame...)
Affinity DataIC50: 2.30nMAssay Description:Antagonist activity against human glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of glucagon-induced glucagon receptor-mediated cAMP production in rat hepatocytes after 15 mins by cAMP dynamic2 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057824(CHEMBL3326175)
Affinity DataIC50: 87nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057820(CHEMBL3326174)
Affinity DataIC50: 160nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057813(CHEMBL3326173)
Affinity DataIC50: 270nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50: 292nMAssay Description:Inhibition of glucagon-induced glucagon receptor-mediated cAMP production in human hepatocytes after 15 mins by cAMP dynamic2 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057806(CHEMBL3326172)
Affinity DataIC50: 430nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057798(CHEMBL3326170)
Affinity DataIC50: 970nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of GLP-1R (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057800(CHEMBL3326171)
Affinity DataIC50: 1.40E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057864(CHEMBL3325456)
Affinity DataIC50: 2.90E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057817(CHEMBL3326187)
Affinity DataIC50: 5.50E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057825(CHEMBL3326176)
Affinity DataIC50: 9.50E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057797(CHEMBL3326165)
Affinity DataIC50: 9.50E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50: 9.60E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057831(CHEMBL3326177)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50058003(CHEMBL3326186)
Affinity DataIC50: 2.40E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057859(CHEMBL3326181)
Affinity DataIC50: 2.70E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057863(CHEMBL3326185)
Affinity DataIC50: 4.40E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057861(CHEMBL3326183)
Affinity DataIC50: 6.90E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057834(CHEMBL3326178)
Affinity DataIC50: 8.90E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057860(CHEMBL3326182)
Affinity DataIC50: 9.30E+4nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057849(CHEMBL3326180)
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057836(CHEMBL3326179)
Affinity DataIC50: 1.80E+5nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057862(CHEMBL3326184)
Affinity DataIC50: 2.70E+5nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed