Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50045341
TargetThromboxane A2 receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50058027(CHEMBL29374)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human TP receptor expressed in QBI-HEK 293A cells assessed as IP3 metabolite level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50058026(CHEMBL3326602)
Affinity DataIC50: 54nMAssay Description:Inhibition of human TP receptor expressed in QBI-HEK 293A cells assessed as IP3 metabolite level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353640(CHEMBL65121)
Affinity DataIC50: 190nMAssay Description:Inhibition of human TP receptor expressed in QBI-HEK 293A cells assessed as IP3 metabolite level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50058025(CHEMBL3326603)
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of human TP receptor expressed in QBI-HEK 293A cells assessed as IP3 metabolite level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed