Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50044666
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024580BDBM50024580(CHEMBL3330612)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at human 5HT1AR expressed in CHO cells assessed as increase in [35S]GTPgammaS binding by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 86757BDBM86757(NSC_11603174 | CAS_0 | [11C]MMP)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at human 5HT1AR expressed in CHO cells assessed as increase in [35S]GTPgammaS binding by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 86757BDBM86757(NSC_11603174 | CAS_0 | [11C]MMP)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024574BDBM50024574(CHEMBL3330616)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024574BDBM50024574(CHEMBL3330616)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human 5HT1AR expressed in CHO cells assessed as increase in [35S]GTPgammaS binding by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024605BDBM50024605(US9290463, E | CHEMBL3330603)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at human 5HT1AR expressed in CHO cells assessed as increase in [35S]GTPgammaS binding by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024567BDBM50024567(CHEMBL3330623)
Affinity DataKi:  0.440nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024643BDBM50024643(CHEMBL3329234)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024647BDBM50024647(CHEMBL3330599)
Affinity DataKi:  0.660nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024577BDBM50024577(CHEMBL3330614)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at human 5HT1AR expressed in CHO cells assessed as increase in [35S]GTPgammaS binding by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024646BDBM50024646(CHEMBL3330600)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024595BDBM50024595(CHEMBL3330605)
Affinity DataKi:  0.835nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024580BDBM50024580(CHEMBL3330612)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024577BDBM50024577(CHEMBL3330614)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024573BDBM50024573(US9290463, A | CHEMBL3330617)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024584BDBM50024584(CHEMBL3330609)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024582BDBM50024582(CHEMBL3330611)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024566BDBM50024566(CHEMBL3330624)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024605BDBM50024605(US9290463, E | CHEMBL3330603)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024583BDBM50024583(CHEMBL3330610)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024587BDBM50024587(CHEMBL3330606)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024575BDBM50024575(CHEMBL3330615)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024585BDBM50024585(CHEMBL3330608)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024603BDBM50024603(US9290463, C | CHEMBL3330604)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024578BDBM50024578(CHEMBL3330613)
Affinity DataKi:  68nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024568BDBM50024568(CHEMBL3330622)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024564BDBM50024564(CHEMBL3330626)
Affinity DataKi:  175nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024576BDBM50024576(Eptapirone)
Affinity DataKi:  175nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024571BDBM50024571(CHEMBL3330619)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024645BDBM50024645(CHEMBL3330601)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024648BDBM50024648(CHEMBL3330598)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024586BDBM50024586(CHEMBL3330607)
Affinity DataKi:  215nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024644BDBM50024644(CHEMBL3330602)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024572BDBM50024572(CHEMBL3330618)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024565BDBM50024565(CHEMBL3330625)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024569BDBM50024569(CHEMBL3330621)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024570BDBM50024570(CHEMBL3330620)
Affinity DataKi:  350nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Stony Brook University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024650BDBM50024650(CHEMBL3330597)
Affinity DataKi:  414nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed