Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50044690
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026204BDBM50026204(CHEMBL3338188)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026071BDBM50026071(CHEMBL3338182)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026077BDBM50026077(CHEMBL3338176)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026202BDBM50026202(CHEMBL3338187)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026236BDBM50026236(CHEMBL3338190)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026239BDBM50026239(CHEMBL3338193)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026235BDBM50026235(CHEMBL3338189)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026240BDBM50026240(CHEMBL3338194)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026176BDBM50026176(CHEMBL3338174)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026237BDBM50026237(CHEMBL3338191)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026072BDBM50026072(CHEMBL3338181)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026238BDBM50026238(CHEMBL3338192)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026177BDBM50026177(CHEMBL3338173)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026068BDBM50026068(CHEMBL3338185)
Affinity DataEC50:  31nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026075BDBM50026075(CHEMBL3338178)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026076BDBM50026076(CHEMBL3338177)
Affinity DataEC50:  37nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026175BDBM50026175(CHEMBL3338175)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026181BDBM50026181(CHEMBL3338169)
Affinity DataEC50:  57nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026074BDBM50026074(CHEMBL3338179)
Affinity DataEC50:  63nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026073BDBM50026073(CHEMBL3338180)
Affinity DataEC50:  95nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026180BDBM50026180(CHEMBL3338170)
Affinity DataEC50:  104nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026178BDBM50026178(CHEMBL3338172)
Affinity DataEC50:  117nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026190BDBM50026190(CHEMBL3338168)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026194BDBM50026194(CHEMBL3338165)
Affinity DataEC50:  133nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026191BDBM50026191(CHEMBL3338167)
Affinity DataEC50:  183nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026179BDBM50026179(CHEMBL3338171)
Affinity DataEC50:  724nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026195BDBM50026195(CHEMBL3338164)
Affinity DataEC50:  1.09E+3nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026240BDBM50026240(CHEMBL3338194)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026201BDBM50026201(CHEMBL3338159)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026192BDBM50026192(CHEMBL3338166)
Affinity DataEC50:  3.50E+3nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026192BDBM50026192(CHEMBL3338166)
Affinity DataEC50:  3.50E+3nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026200BDBM50026200(CHEMBL3338160)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026198BDBM50026198(CHEMBL3338162)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026199BDBM50026199(CHEMBL3338161)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026196BDBM50026196(CHEMBL3338163)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026070BDBM50026070(CHEMBL3338183)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026069BDBM50026069(CHEMBL3338184)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026067BDBM50026067(CHEMBL3338186)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026072BDBM50026072(CHEMBL3338181)
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of PXR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Departments of Discovery Chemistry, Metabolic Diseases, Lead Evaluation, Computer-Assisted Drug Design, Discovery Toxicology, Exploratory Clinical and Translational Research, and Pharmaceutical Candi

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026240BDBM50026240(CHEMBL3338194)
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of PXR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed