Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 6814
TargetDipeptidyl peptidase 4(Human)
Csir-Central Drug Research Institute

LigandPNGBDBM11162(Triazolopiperazine Analogue 1 | (3R)-3-amino-1-[3-...)
Affinity DataIC50: 18nMAssay Description:DPP-IV inhibitory activity was determined by measuring the p-nitroaniline (pNA) released from the chromogenic substrate hydrolysis (H-Gly-Pro-pNA). T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2015
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Csir-Central Drug Research Institute

LigandPNGBDBM152800(1-(2-(4-(7-Chloro-4-quinolyl)piperazin-1-yl)acetyl...)
Affinity DataIC50: 3.73E+3nMAssay Description:DPP-IV inhibitory activity was determined by measuring the p-nitroaniline (pNA) released from the chromogenic substrate hydrolysis (H-Gly-Pro-pNA). T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2015
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Csir-Central Drug Research Institute

LigandPNGBDBM152801(4-(2-(4-(7-Chloro-4-quinolyl)piperazin-1-yl)acetyl...)
Affinity DataIC50: 5.96E+3nMAssay Description:DPP-IV inhibitory activity was determined by measuring the p-nitroaniline (pNA) released from the chromogenic substrate hydrolysis (H-Gly-Pro-pNA). T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2015
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Csir-Central Drug Research Institute

LigandPNGBDBM152799(1-(2-(4-(3-chlorophenyl)piperazin-1-yl)acetyl)pipe...)
Affinity DataIC50: 6.06E+3nMAssay Description:DPP-IV inhibitory activity was determined by measuring the p-nitroaniline (pNA) released from the chromogenic substrate hydrolysis (H-Gly-Pro-pNA). T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2015
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Csir-Central Drug Research Institute

LigandPNGBDBM152798(3-(2-(4-(2-Pyridyl)piperazin-1-yl)acetyl)thiazolid...)
Affinity DataIC50: 6.08E+3nMAssay Description:DPP-IV inhibitory activity was determined by measuring the p-nitroaniline (pNA) released from the chromogenic substrate hydrolysis (H-Gly-Pro-pNA). T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2015
Entry Details Article
PubMed