Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50006169
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497521(CHEMBL3337749)
Affinity DataIC50: 190nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497538(CHEMBL3337748)
Affinity DataIC50: 230nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497533(CHEMBL3337746)
Affinity DataIC50: 400nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497531(CHEMBL3337750)
Affinity DataIC50: 670nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497532(CHEMBL3337751)
Affinity DataIC50: 700nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497517(CHEMBL3337739)
Affinity DataIC50: 700nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497528(CHEMBL3337742)
Affinity DataIC50: 720nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497520(CHEMBL3337747)
Affinity DataIC50: 800nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497525(CHEMBL3337744)
Affinity DataIC50: 830nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497527(CHEMBL3337741)
Affinity DataIC50: 840nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497522(CHEMBL186008)
Affinity DataIC50: 980nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497538(CHEMBL3337748)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497518(CHEMBL3337738)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497519(CHEMBL3337745)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497529(CHEMBL3337743)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497536(CHEMBL3337629)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497530(CHEMBL3337638)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497523(CHEMBL3337736)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497521(CHEMBL3337749)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497528(CHEMBL3337742)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497537(CHEMBL3337628)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497535(CHEMBL3337630)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497527(CHEMBL3337741)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497526(CHEMBL3337737)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497528(CHEMBL3337742)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497524(CHEMBL3245455)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497540(CHEMBL3245452)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497520(CHEMBL3337747)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497527(CHEMBL3337741)
Affinity DataIC50: 1.29E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497533(CHEMBL3337746)
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497517(CHEMBL3337739)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497517(CHEMBL3337739)
Affinity DataIC50: 1.62E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497525(CHEMBL3337744)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497525(CHEMBL3337744)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497531(CHEMBL3337750)
Affinity DataIC50: 1.88E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497532(CHEMBL3337751)
Affinity DataIC50: 1.89E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497519(CHEMBL3337745)
Affinity DataIC50: 1.89E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497533(CHEMBL3337746)
Affinity DataIC50: 1.97E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497530(CHEMBL3337638)
Affinity DataIC50: 2.34E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497523(CHEMBL3337736)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497530(CHEMBL3337638)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497523(CHEMBL3337736)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497522(CHEMBL186008)
Affinity DataIC50: 3.01E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497518(CHEMBL3337738)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497529(CHEMBL3337743)
Affinity DataIC50: 4.21E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497518(CHEMBL3337738)
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497539(CHEMBL3337631)
Affinity DataIC50: 4.55E+4nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase(Staphylococcus aureus (strain MW2))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497526(CHEMBL3337737)
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497526(CHEMBL3337737)
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50497529(CHEMBL3337743)
Affinity DataIC50: 5.37E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
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