Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 6745
TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))
Affinity DataIC50: 150nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2015
Entry Details Article
PubMed
TargetDeath-associated protein kinase 1(Human)
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))
Affinity DataKd:  240nMpH: 7.5Assay Description:40 µL of a solution containing 350-500 µM of CPR005231 (compound 6) were titrated into the 200 µL sample cell containing 25-55 µM DAPK1 (AA 1-285) or...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2015
Entry Details Article
PubMed
TargetDeath-associated protein kinase 1(Human)
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))
Affinity DataIC50: 247nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))
Affinity DataIC50: 1.60E+3nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2015
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))
Affinity DataIC50: 1.80E+3nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 5(Human)
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))
Affinity DataIC50: 5.60E+3nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2015
Entry Details Article
PubMed