Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50006192
LigandChemical structure of BindingDB Monomer ID 50030474BDBM50030474(US9562012, rosiglitazone | CHEBI:50122 | Avandamet...)
Affinity DataEC50:  1.60E+3nMAssay Description:Transactivation of PPAR transfected in human HepG2 cells after 20 hrs by PPAR-luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 50497669BDBM50497669(CHEMBL3353021)
Affinity DataEC50:  6.40E+3nMAssay Description:Transactivation of PPAR transfected in human HepG2 cells after 20 hrs by PPAR-luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497670BDBM50497670(CHEMBL3353020)
Affinity DataEC50:  8.20E+3nMAssay Description:Transactivation of PPAR transfected in human HepG2 cells after 20 hrs by PPAR-luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497663BDBM50497663(CHEMBL3353023)
Affinity DataEC50:  1.87E+4nMAssay Description:Transactivation of PPAR transfected in human HepG2 cells after 20 hrs by PPAR-luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497664BDBM50497664(CHEMBL3353024)
Affinity DataEC50:  2.06E+4nMAssay Description:Transactivation of PPAR transfected in human HepG2 cells after 20 hrs by PPAR-luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497672BDBM50497672(CHEMBL3353025)
Affinity DataEC50:  2.23E+4nMAssay Description:Transactivation of PPAR transfected in human HepG2 cells after 20 hrs by PPAR-luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497667BDBM50497667(CHEMBL3353026)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of PPAR transfected in human HepG2 cells after 20 hrs by PPAR-luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497666BDBM50497666(CHEMBL3353027)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of PPAR transfected in human HepG2 cells after 20 hrs by PPAR-luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497668BDBM50497668(CHEMBL3353022)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of PPAR transfected in human HepG2 cells after 20 hrs by PPAR-luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497665BDBM50497665(CHEMBL3353030)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of PPAR transfected in human HepG2 cells after 20 hrs by PPAR-luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497671BDBM50497671(CHEBI:64976 | CHEMBL3353029)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of PPAR transfected in human HepG2 cells after 20 hrs by PPAR-luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50497673BDBM50497673(CHEMBL3353028)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of PPAR transfected in human HepG2 cells after 20 hrs by PPAR-luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed