Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50044967
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50035131BDBM50035131((1S,9S,13S)-1,13-dimethyl-10-(3-methylbut-2-enyl)-...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50299706BDBM50299706(4-Cyclohexyl-1-[3-(5-methoxy-1,2,3,4-tetrahydronap...)
Affinity DataKi:  143nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353279BDBM50353279(CHEMBL1830683 | CHEMBL259582)
Affinity DataKi:  151nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50038697BDBM50038697(CHEMBL3354875)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50038704BDBM50038704(CHEMBL3354882)
Affinity DataKi:  1.39E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50038726BDBM50038726(CHEMBL3354886)
Affinity DataKi:  2.19E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50038698BDBM50038698(CHEMBL3354877)
Affinity DataKi:  2.93E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50038701BDBM50038701(CHEMBL3354879)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50038702BDBM50038702(CHEMBL3354880)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50038700BDBM50038700(CHEMBL3354878)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50038699BDBM50038699(CHEMBL3352842)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50038727BDBM50038727(CHEMBL3354887)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50038728BDBM50038728(CHEMBL3354888)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50038725BDBM50038725(CHEMBL3354885)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50038722BDBM50038722(CHEMBL3354883)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50038724BDBM50038724(CHEMBL3354884)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50038703BDBM50038703(CHEMBL3354881)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed