Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 4753
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM26263(ethyl 12-fluoro-8-methyl-9-oxo-2,4,8-triazatricycl...)
Affinity DataKi:  0.480nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM26263(ethyl 12-fluoro-8-methyl-9-oxo-2,4,8-triazatricycl...)
Affinity DataKi:  0.490nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM26263(ethyl 12-fluoro-8-methyl-9-oxo-2,4,8-triazatricycl...)
Affinity DataKi:  0.620nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM26263(ethyl 12-fluoro-8-methyl-9-oxo-2,4,8-triazatricycl...)
Affinity DataKi:  0.720nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM50243981(CHEMBL453066 | Beta CCM | Methyl Beta-carboline-3 ...)
Affinity DataKi:  0.780nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM26263(ethyl 12-fluoro-8-methyl-9-oxo-2,4,8-triazatricycl...)
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM26263(ethyl 12-fluoro-8-methyl-9-oxo-2,4,8-triazatricycl...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM50019213(5-(2-chlorophenyl)-7-nitro-1,3-dihydro-2H-1,4-benz...)
Affinity DataKi:  1.27nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM50019213(5-(2-chlorophenyl)-7-nitro-1,3-dihydro-2H-1,4-benz...)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM50019213(5-(2-chlorophenyl)-7-nitro-1,3-dihydro-2H-1,4-benz...)
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM50243981(CHEMBL453066 | Beta CCM | Methyl Beta-carboline-3 ...)
Affinity DataKi:  2.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM50243981(CHEMBL453066 | Beta CCM | Methyl Beta-carboline-3 ...)
Affinity DataKi:  4.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM81951(NSC_104999 | CAS_104999 | DMCM)
Affinity DataKi:  5.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGamma-aminobutyric acid receptor subunit alpha-3(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM81951(NSC_104999 | CAS_104999 | DMCM)
Affinity DataKi:  10.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM81951(NSC_104999 | CAS_104999 | DMCM)
Affinity DataKi:  14.4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)
Affinity DataKi:  16.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGamma-aminobutyric acid receptor subunit alpha-2(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)
Affinity DataKi:  16.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGamma-aminobutyric acid receptor subunit alpha-3(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)
Affinity DataKi:  17nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM50026756(CHEMBL13662 | CL 218872 | 3-Methyl-6-(3-trifluorom...)
Affinity DataKi:  108nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM81952(NSC_93250 | CAS_93250 | 2-Oxoquazepam)
Affinity DataKi:  205nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM81952(NSC_93250 | CAS_93250 | 2-Oxoquazepam)
Affinity DataKi:  236nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM50026756(CHEMBL13662 | CL 218872 | 3-Methyl-6-(3-trifluorom...)
Affinity DataKi:  405nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM50026756(CHEMBL13662 | CL 218872 | 3-Methyl-6-(3-trifluorom...)
Affinity DataKi:  1.62E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM50026756(CHEMBL13662 | CL 218872 | 3-Methyl-6-(3-trifluorom...)
Affinity DataKi:  1.74E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM50026756(CHEMBL13662 | CL 218872 | 3-Methyl-6-(3-trifluorom...)
Affinity DataKi:  1.79E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Human)
UniversitÄT Heidelberg

Curated by PDSP Ki Database
LigandPNGBDBM50026756(CHEMBL13662 | CL 218872 | 3-Methyl-6-(3-trifluorom...)
Affinity DataKi:  2.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed