Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50045048
TargetMaternal embryonic leucine zipper kinase(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50043341(CHEMBL3355059)
Affinity DataIC50: 37nMAssay Description:Inhibition of MELK kinase (unknown origin) using biotinylated ZIP-tide peptide/gamma[33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetMaternal embryonic leucine zipper kinase(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50043342(CHEMBL3355058)
Affinity DataIC50: 410nMAssay Description:Inhibition of MELK kinase (unknown origin) using biotinylated ZIP-tide peptide/gamma[33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetMaternal embryonic leucine zipper kinase(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50043345(CHEMBL3355056)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of MELK kinase (unknown origin) using biotinylated ZIP-tide peptide/gamma[33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetMaternal embryonic leucine zipper kinase(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50043325(CHEMBL3355054)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of MELK kinase (unknown origin) using biotinylated ZIP-tide peptide/gamma[33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetMaternal embryonic leucine zipper kinase(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50043369(CHEMBL3355055)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of MELK kinase (unknown origin) using biotinylated ZIP-tide peptide/gamma[33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50043341(CHEMBL3355059)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of Flt3 (unknown origin) by Millipore kinase analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetMaternal embryonic leucine zipper kinase(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50043341(CHEMBL3355059)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of MELK kinase (unknown origin) using KKLNRTLSFAEPG/gamma[33P]ATP by Millipore kinase/scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetMaternal embryonic leucine zipper kinase(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50043344(CHEMBL3355057)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of MELK kinase (unknown origin) using biotinylated ZIP-tide peptide/gamma[33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMaternal embryonic leucine zipper kinase(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50043333(CHEMBL3355053)
Affinity DataIC50: 1.60E+5nMAssay Description:Inhibition of MELK kinase (unknown origin) using biotinylated ZIP-tide peptide/gamma[33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50043341(CHEMBL3355059)
Affinity DataIC50: 7.60E+5nMAssay Description:Inhibition of Mnk2 (unknown origin) by Millipore kinase analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
LigandPNGBDBM50043341(CHEMBL3355059)
Affinity DataIC50: 8.10E+5nMAssay Description:Inhibition of CAMK2delta (unknown origin) by Millipore kinase analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
LigandPNGBDBM50043341(CHEMBL3355059)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of CAMK2gamma (unknown origin) by Millipore kinase analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetMyosin light chain kinase, smooth muscle(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50043341(CHEMBL3355059)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of MLCK (unknown origin) by Millipore kinase analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed