TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 4.50E+3nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.54E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase Y181C mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.59E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase L100I mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 2.00E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase G190A mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 6.33E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 6.76E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 6.99E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataIC50: 1.21E+4nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataIC50: 1.57E+4nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataIC50: 4.45E+4nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataIC50: 6.29E+4nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataIC50: 6.88E+4nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataIC50: 7.93E+4nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataIC50: 1.14E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataIC50: 1.49E+5nMAssay Description:Inhibition of HIV1 ribonuclease H pre-incubated with compound before enzyme addition using using RNA/DNA heteroduplex and measured after 60 mins by p...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataIC50: 1.94E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataIC50: 2.11E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair