Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50046239
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of ALK (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of ALK (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of ALK (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of ALK (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of ALK (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of ALK (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of ALK (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of ALK (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of ALK (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of ALK (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of ALK (unknown origin) by cellular assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of ALK (unknown origin) by cellular assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of ALK (unknown origin) by cellular assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of ALK (unknown origin) by cellular assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of ALK (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of ALK (unknown origin) by cellular assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of ALK (unknown origin) by cellular assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of ALK (unknown origin) by cellular assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of ALK (unknown origin) by cellular assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of ALK (unknown origin) by cellular assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of human ERG by patch clamp cellular assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Teva Branded Pharmaceutical Products R & D
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG by patch clamp cellular assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2D6A (unknown origin)More data for this Ligand-Target Pair










