Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50045709
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077906BDBM50077906(CHEMBL3305901)
Affinity DataKd:  0.480nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077906BDBM50077906(CHEMBL3305901)
Affinity DataKi:  0.550nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077924BDBM50077924(CHEMBL3417124)
Affinity DataKi:  1.20nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077980BDBM50077980(CHEMBL3417117)
Affinity DataKi:  1.60nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077991BDBM50077991(CHEMBL3417237)
Affinity DataKi:  2nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077912BDBM50077912(CHEMBL3417231)
Affinity DataKi:  2nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077986BDBM50077986(CHEMBL3417111)
Affinity DataKi:  2.20nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077972BDBM50077972(CHEMBL3417118)
Affinity DataKi:  2.30nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077908BDBM50077908(CHEMBL3417235)
Affinity DataKi:  2.40nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077913BDBM50077913(CHEMBL3417230)
Affinity DataKi:  3.40nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077966BDBM50077966(CHEMBL3417119)
Affinity DataKi:  4.40nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077911BDBM50077911(CHEMBL3417232)
Affinity DataKi:  4.5nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077984BDBM50077984(CHEMBL3417113)
Affinity DataKi:  4.60nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077990BDBM50077990(CHEMBL3417238)
Affinity DataKi:  4.60nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077981BDBM50077981(CHEMBL3417116)
Affinity DataKi:  4.90nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077925BDBM50077925(CHEMBL3417123)
Affinity DataKi:  7.90nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077918BDBM50077918(CHEMBL3417225)
Affinity DataKi:  10nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077916BDBM50077916(CHEMBL3417227)
Affinity DataKi:  10nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077921BDBM50077921(CHEMBL3417221)
Affinity DataKi:  11nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077914BDBM50077914(CHEMBL3417229)
Affinity DataKi:  12nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077926BDBM50077926(CHEMBL3417122)
Affinity DataKi:  13nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077950BDBM50077950(CHEMBL3417120)
Affinity DataKi:  13nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077910BDBM50077910(CHEMBL3417233)
Affinity DataKi:  13nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077987BDBM50077987(CHEMBL3417110)
Affinity DataKi:  15nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077983BDBM50077983(CHEMBL3417114)
Affinity DataKi:  15nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077982BDBM50077982(CHEMBL3417115)
Affinity DataKi:  21nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077948BDBM50077948(CHEMBL3417121)
Affinity DataKi:  23nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077915BDBM50077915(CHEMBL3417228)
Affinity DataKi:  23nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077907BDBM50077907(CHEMBL3417236)
Affinity DataKi:  24nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077985BDBM50077985(CHEMBL3417112)
Affinity DataKi:  31nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077920BDBM50077920(CHEMBL3417223)
Affinity DataKi:  39nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077917BDBM50077917(CHEMBL3417226)
Affinity DataKi:  41nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077923BDBM50077923(CHEMBL3417216)
Affinity DataKi:  49nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257992BDBM50257992((1S,3R)-N-(3,5-bis(trifluoromethyl)benzyl)-3-(2,3-...)
Affinity DataKi:  50nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077922BDBM50077922(CHEMBL3417220)
Affinity DataKi:  55nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077919BDBM50077919(CHEMBL3417224)
Affinity DataKi:  75nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077909BDBM50077909(CHEMBL3417234)
Affinity DataKi:  83nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077988BDBM50077988(CHEMBL3417240)
Affinity DataKi:  137nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Leiden University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50077989BDBM50077989(CHEMBL3417239)
Affinity DataKi:  199nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMed