Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50045485
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064422BDBM50064422(CHEMBL3401162)
Affinity DataIC50: 25nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064422BDBM50064422(CHEMBL3401162)
Affinity DataKi:  40nMAssay Description:Irreversible inhibition of rat hormone sensitive lipase assessed as relative residual activity by kinetic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064413BDBM50064413(CHEMBL3401168)
Affinity DataIC50: 60nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064423BDBM50064423(CHEMBL3401161)
Affinity DataIC50: 75nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064414BDBM50064414(CHEMBL3401167)
Affinity DataIC50: 360nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064421BDBM50064421(CHEMBL3401163)
Affinity DataIC50: 420nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064418BDBM50064418(CHEMBL3401164)
Affinity DataIC50: 450nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064416BDBM50064416(CHEMBL3401165)
Affinity DataIC50: 470nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064425BDBM50064425(CHEMBL3401160)
Affinity DataIC50: 900nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064415BDBM50064415(CHEMBL3401166)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064408BDBM50064408(CHEMBL3401171)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064410BDBM50064410(CHEMBL3401170)
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064427BDBM50064427(CHEMBL3401172)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064411BDBM50064411(CHEMBL2179369)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064409BDBM50064409(CHEMBL2179367)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50308520BDBM50308520(cyclophostin | CHEMBL603622)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50308513BDBM50308513((3R,8aR)-3-Methoxy-5-methyl-3-oxo-8,8a-dihydro-1H-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064428BDBM50064428(CHEMBL2179365)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064412BDBM50064412(CHEMBL3401169)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Rat)
University of Missouri St. Louis

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064426BDBM50064426(CHEMBL3401159)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed