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Found 24 Enz. Inhib. hit(s) with all data for entry = 50045453
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063062(CHEMBL3398394)
Affinity DataIC50:  205nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063060(CHEMBL3398391)
Affinity DataIC50:  247nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063061(CHEMBL3398392)
Affinity DataIC50:  253nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063058(CHEMBL3398389)
Affinity DataIC50:  329nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50380061(CHEMBL2012637)
Affinity DataIC50:  360nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063055(CHEMBL3398398)
Affinity DataIC50:  433nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063055(CHEMBL3398398)
Affinity DataIC50:  463nMAssay Description:Displacement of [3H]Mesulergine from human recombinant 5-HT2C receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063063(CHEMBL3398395)
Affinity DataIC50:  479nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063061(CHEMBL3398392)
Affinity DataIC50:  480nMAssay Description:Displacement of [3H]Mesulergine from human recombinant 5-HT2C receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063065(CHEMBL3398397)
Affinity DataIC50:  555nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063059(CHEMBL3398390)
Affinity DataIC50:  702nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063062(CHEMBL3398394)
Affinity DataIC50:  740nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063062(CHEMBL3398394)
Affinity DataIC50:  1.04E+3nMAssay Description:Displacement of [3H]Mesulergine from human recombinant 5-HT2C receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063063(CHEMBL3398395)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063064(CHEMBL3398396)
Affinity DataIC50:  1.59E+3nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063058(CHEMBL3398389)
Affinity DataIC50:  1.83E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063056(CHEMBL2414732)
Affinity DataIC50:  2.04E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063061(CHEMBL3398392)
Affinity DataIC50:  2.12E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063064(CHEMBL3398396)
Affinity DataIC50:  2.44E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063055(CHEMBL3398398)
Affinity DataIC50:  2.53E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063065(CHEMBL3398397)
Affinity DataIC50:  2.96E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063057(CHEMBL3398399)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063059(CHEMBL3398390)
Affinity DataIC50:  4.97E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063060(CHEMBL3398391)
Affinity DataIC50:  6.34E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed